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2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(pyridin-2-ylmethyl)acetamide
4-chloro-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1-methyl-1H-pyrazole-3-carboxamide
[2-(4,6-dimethylpyrimidin-2-yl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-(5-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
1-(2-{2-ethyl-4-[(propan-2-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)pyrrolidin-2-one
1-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N,1-diethyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
(5-{[3-(2-phenylethyl)piperidin-1-yl]methyl}furan-2-yl)methanol
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1-(pyrimidin-2-yl)piperidin-4-amine
2-cyclopropyl-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
7-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]piperidine-4-carboxamide
2-ethyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}pyrimidine-5-carboxamide
1-ethyl-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-ethyl-4-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
5-amino-3-[5-(oxolan-2-yl)thiophen-2-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
8-[(3-ethoxy-2-hydroxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-oxoethyl)urea
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}urea
N-cyclooctyl-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclopropanecarbonyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
3-{2-[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
N-({7-[2-(3-chlorophenoxy)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-methylfuran-3-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-3-(pyridin-4-yl)propanamide
(3S,4R)-1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
2-{[(cyclopropylmethyl)(2-methoxyethyl)amino]methyl}-6-fluoroquinolin-4-ol
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-benzothiazole
1-(cyclohexylmethyl)-2-(methoxymethyl)-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
N-cyclopentyl-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(3aS,6aR)-5-(2,3-dihydro-1H-inden-2-yl)-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-(1-{1-[(2R)-2-amino-4,4-dimethylpentanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
(1-{2-[(5-ethylpyrimidin-2-yl)amino]ethyl}piperidin-3-yl)methanol
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
4-(furan-2-yl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-5-propyl-1,2-oxazole-3-carboxamide
N3-(2-methoxyethyl)-N5-[(1R)-1-(4-methoxyphenyl)ethyl]-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-cyclopentyl-3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]piperidine
methyl 3-({5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propanoate
N-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(2E)-1-{3-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxymethyl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
2-(2-methoxy-4-methylphenoxymethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-(methylamino)-1,3-thiazole-4-carboxamide
2-(1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)ethan-1-amine
1-[1-(2-chloro-4-fluorobenzoyl)piperidin-3-yl]-2-phenylethan-1-one