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7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-(quinoline-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethyl)piperidine-4-carboxylate
3-ethyl-1-[3-(3-methoxyphenyl)propanoyl]piperidine-3-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
5-ethyl-2,3-dimethyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-methyl-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
(3S,4S)-1-(2-amino-6-methylpyrimidin-4-yl)-4-(propan-2-yloxy)pyrrolidin-3-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(2-methylpropanesulfonyl)ethyl]acetamide
4-[(4-methoxy-3-methylphenyl)methyl]-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-[(methylsulfanyl)methyl]-5-[4-(1H-pyrazol-3-yl)phenyl]-1,2,4-oxadiazole
3-butanamido-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylbenzamide
(3S,4R)-N,N-dimethyl-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-(propan-2-yl)pyrrolidin-3-amine
N,N-dimethyl-2-(4-{5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}piperazin-1-yl)acetamide
5-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(4-methyl-1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-4-(2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzoyl)-1,3-dimethylpiperazin-2-one
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(4-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,N-dimethyl-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}azepan-4-amine
(2S,4R)-4-[(1,3-benzoxazol-2-yl)amino]-N-methyl-1-(pentan-3-yl)pyrrolidine-2-carboxamide
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-3-phenoxypropan-1-one
methyl 3-(2-methylpropanamido)-6-(thiomorpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
N-(adamantan-1-yl)-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl 9-(cyclopentyloxy)-3-{[3-(2-hydroxyethoxy)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-butyl-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
9-[(2-ethylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[1-(2-methoxybenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylthiophene-3-carboxamide
2-methoxy-N-(1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-phenylpropanamide
8-[(5-fluoro-2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-(naphthalen-2-ylmethyl)-2,7-diazaspiro[4.5]decane
methyl 4-(5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N,N-diethyl-2-{4-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
1-(2-{[(2E)-3,7-dimethylocta-2,6-dien-1-yl]amino}ethyl)cyclopentan-1-ol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methylphenyl)acetamide
2-(3-methoxypropyl)-8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-(dimethylamino)ethyl]-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
7-[2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-ethoxy-4-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazol-2-yl]phenol
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(1,3-thiazol-2-yl)piperazin-2-yl}ethan-1-ol
5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
1-(1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
ethyl 4-(2-phenoxyethyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxylate
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-4H-chromen-4-one
[3-(2-methylquinazolin-4-yl)phenyl]methanol
1-(2-phenylethyl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-oxo-2-phenylacetamide
(4aS,7aR)-1-[(4-fluoro-3-methylphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione