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4-[2-(3,4-dimethoxyphenyl)acetyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
1-{2-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]phenyl}ethan-1-one
[(3R,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(furan-2-ylmethyl)({[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl})(prop-2-yn-1-yl)amine
8-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-(quinolin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2-{[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
1-propyl-4-{4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}pyrrolidin-2-one
1-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-3-(prop-2-en-1-yl)urea
N-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-6-fluoro-N-methylquinoline-4-carboxamide
{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
3-(3,4-dimethylphenyl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
(1S,6R)-3-methyl-9-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(2S,4R,6S)-2-benzyl-6-(4-chlorophenyl)oxan-4-yl]acetamide
N-methyl-2-[2-(methylsulfanyl)acetyl]-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(1S,3R)-3-amino-N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)cyclopentane-1-carboxamide
(2E)-N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-fluorophenyl)prop-2-enamide
N-[(3R,4S)-4-cyclopropyl-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-yl]methanesulfonamide
1-{2-[1-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
3-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
3,3-dimethyl-1-[(3S,4R)-1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea
2-({[(3R,4R)-1-(4-chloro-2-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-methyl-1'-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
[(3R,5R)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
9-[(2R)-2-amino-2-cyclohexylacetyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-5-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazole
2-(4-chlorophenyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}morpholine
1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]-2-phenylethan-1-one
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-(quinolin-6-yl)urea
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclohexyl-4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-5-(2-methoxyethyl)-1H-1,2,4-triazole
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-(methylsulfanyl)acetamide
N-(3-methanesulfonamidophenyl)-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
(4aS,7aR)-1-[(3-methoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
5-{4-[(2,4-difluorophenyl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
1-methyl-N-{[4-(2-methylpropoxy)phenyl]methyl}-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
2-(3,4-dichlorophenyl)-4-(2-methoxy-3-methylbenzoyl)morpholine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-3-hydroxypyridine-2-carboxamide
(1S,5R)-6-benzyl-3-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 3-(furan-2-amido)-5-({[3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}methyl)benzoate
1-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-amine
1-(4-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-4-oxobutyl)piperidin-2-one
2-(2-fluorophenoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
1-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
5-[1-(pent-4-enoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-benzyl-N,5-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide