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{4-benzyl-1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}methanol
1'-(3-methyl-1,2-oxazole-5-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({1-[(2-chlorophenyl)methyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
4-(2,6-difluorophenoxy)-1-(hexan-2-yl)piperidine-4-carboxylic acid
N-methyl-2-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}propanamide
7-[2-(1H-pyrazol-1-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1,8-bis(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-ethyl-2-methyl-1H-indol-5-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-{1-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
3-[3-oxo-4-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepane-1-carbonyl]pyridin-1-ium-1-olate
5-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[5-(methylcarbamoyl)thiophen-2-yl]-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
2-[benzyl(methyl)amino]-N-(2-hydroxybutyl)-2,3-dihydro-1H-indene-2-carboxamide
(4-{[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methanol
(1S,4S)-2-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
1-(4-chloro-2-methoxy-5-methylphenyl)-3-(furan-2-ylmethyl)-3-(2-hydroxyethyl)urea
3-methyl-8-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
N-(4-methoxy-2-methylphenyl)-3-[1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]propanamide
ethyl 4-({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)piperidine-1-carboxylate
methyl 4-[(3-{[3-(1H-pyrazol-1-yl)phenyl]carbamoyl}piperidin-1-yl)methyl]benzoate
2-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-fluoropyridine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(1,3-thiazol-4-yl)ethan-1-one
N-{[5-(2-phenylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
(1R,5R)-3-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
3-methyl-5-[4-(1H-pyrazol-5-yl)phenyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-(3-chlorophenoxy)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
N-[1-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylfuran-2-yl)methyl]acetamide
2-fluoro-N-({3-methyl-7-[2-(2,3,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
4-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
6-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
3-cyclopropyl-1-methyl-5-(2,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-[2-(3-phenylpropoxy)phenyl]acetamide
(2R)-1-[3-(piperidin-4-ylmethyl)benzoyl]pyrrolidine-2-carboxamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
N-[3-(4-hydroxyphenyl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
N-[(3S,4R)-4-(propan-2-yl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]methanesulfonamide
4-(5-fluoro-2-methylphenyl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-fluorophenyl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
ethyl 3-benzyl-1-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxylate
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
[(2R)-1-(quinoxaline-6-carbonyl)pyrrolidin-2-yl]methanol
(1R,3S)-7-[5-(ethylsulfanyl)thiophene-2-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
(2R,3R)-3-amino-1'-(5-propyl-1,2-oxazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol