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2-methyl-2-(2-{methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
4-(3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-(3-methoxyphenyl)piperazin-2-one
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(3-methylpyridin-2-yl)piperazine
3,4-dimethoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
[2-(2-{1-[6-(methoxymethyl)pyridine-2-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]dimethylamine
6-[3-(3-hydroxypiperidin-1-yl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[1-(2-hydroxypropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
6-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
6-methyl-4-(2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(3R,4S)-4-[({4-[3-(dimethylamino)propoxy]phenyl}methyl)(methyl)amino]oxolan-3-ol
[5-(1-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
N-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-azabicyclo[2.2.2]octan-3-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(4-hydroxyphenyl)propanamide
1-[(2S)-2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethan-1-one
N-[(2,4-dihydroxyphenyl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-4-(hydroxymethyl)azepan-4-ol
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-1-(propan-2-yl)piperidine-4-carboxamide
1-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
{1-[(4-chlorophenyl)methyl]-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl}methanol
2-{1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[2-(4-fluorophenyl)ethyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
2-(2-phenyl-1H-imidazol-1-yl)-1-(thiomorpholin-4-yl)ethan-1-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(quinolin-4-ylmethyl)piperidin-4-yl]propanamide
5-ethyl-2-[1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]pyridine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-3-(piperidin-3-yl)benzamide
8-(adamantan-2-yl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-chlorophenyl)-4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-5-methylpiperazin-2-one
4-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-3-yl]benzoic acid
6-(4-chlorophenyl)-N-(6-hydroxy-6-methylheptan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(1-methoxybutan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)-N-cyclopentylpropanamide
2-methoxy-N-(1-{3-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-methyl-1-[4-(pyridin-2-ylmethoxy)phenyl]urea
dimethyl({4-[1-(4-methylpiperazine-1-carbonyl)piperidin-2-yl]phenyl}methyl)amine
N-pentyl-N'-(2,4,6-trimethylphenyl)butanediamide
3-(2,1,3-benzothiadiazol-5-ylmethyl)-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-ethyl-6-oxo-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
1-(2-chlorophenyl)-4-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazine
1-(cyclopropylmethyl)-5-(4-methylpentanoyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2R,3R)-3-({2-[methyl(phenyl)amino]ethyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1R,5R)-6-benzyl-3-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-3-yl)methyl]furan-2-carboxamide
4-[1-(4-chlorobenzoyl)piperidin-4-yl]-5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidine
(3R,4R)-1-[(5-cyclohexylthiophen-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
N-[2-(4-fluorophenyl)-2-hydroxyethyl]-2-(1-propylpiperidin-4-yl)acetamide