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N-benzyl-1-cyclopropyl-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
1-(furan-2-ylmethyl)-4-(9H-purin-6-yl)-1,4-diazepan-6-ol
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
1-(2-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-3-(4-hydroxyphenyl)benzamide
N-[2-(diethylamino)ethyl]-N-ethyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
5-chloro-3-[(3-methyl-1H-pyrazol-5-yl)methyl]-3,4-dihydroquinazolin-4-one
N-{[7-(2-ethylbutanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
N-[1-(hydroxymethyl)cyclopentyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
(3R,4R)-4-(azepan-1-yl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-ol
8-[3-(4-carbamoylphenoxy)propyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,4S)-4-amino-N,N-diethyl-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidine-2-carboxamide
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)propanamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-(2,3-difluorophenyl)-N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-(4-fluorophenyl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1,2,3,6-tetrahydropyridine
2-{2-[5-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}carbamoyl)thiophen-2-yl]pyrrolidin-1-yl}acetic acid
1-methyl-4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]imidazolidin-2-one
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(3-fluorophenyl)methyl]piperazine
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}urea
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(oxan-4-ylmethyl)pyrrolidine-3-carboxylic acid
N,4-dimethyl-5-(3-methyl-3-phenylpiperidine-1-carbonyl)-1,3-thiazol-2-amine
6-{3-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
N-cyclopropyl-4-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-imidazole-2-carboxamide
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(propan-2-yloxy)ethan-1-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
4-cyclobutyl-6-methyl-2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidine
methyl (2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-(2-fluorobenzamido)pyrrolidine-2-carboxylate
1-[(diethylcarbamoyl)methyl]-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(pyridine-3-sulfonyl)pyrrolidin-3-yl]acetamide
3-methyl-6-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methoxy}-1,2-benzoxazole
2-(2-hydroxyphenoxy)-N-methyl-N-(oxan-2-ylmethyl)acetamide
3-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
1-[4-(cycloheptylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[(3S)-2-oxoazepan-3-yl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}amine
6-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanamide
4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-5-methyl-1-phenylpiperazin-2-one
3-(1H-1,2,3-benzotriazol-1-yl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]propan-1-one
1-cyclopentyl-4-oxo-N3-(propan-2-yl)-N5-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[2-(hydroxymethyl)pyridin-4-yl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(5-propylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenyl-N-[2-(pyridin-4-yl)ethyl]benzamide