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N-[(3-chloro-1-benzothiophen-2-yl)methyl]-1-cyclohexyl-N-methyl-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-(3-cyclopropylpropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(1-methyl-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)methanol
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-3-carboxamide
3-{1-[(6-hydroxynaphthalen-2-yl)methyl]piperidin-3-yl}propanoic acid
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(oxolane-2-carbonyl)piperidine
11-{[(2,4-difluorophenyl)methyl]amino}-4-[2-(dimethylamino)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(4-chloro-1-ethyl-1H-pyrazole-3-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
3-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
(2S,4S)-1-[(3,4-difluorophenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
1-methyl-5-[methyl(2-methylpropyl)amino]-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-1H-pyrazole-3-carboxylic acid
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(methoxymethyl)furan-2-carboxamide
methyl({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})(1H-pyrazol-5-ylmethyl)amine
2-{1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl}benzoic acid
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-4-yl)ethyl]amine
N-(2,5-dimethylphenyl)-3-({6-methylpyrazolo[1,5-a]pyrimidin-3-yl}formamido)propanamide
3-(1H-imidazole-5-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
N-methyl-N-{3-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]propyl}aniline
2-[4-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)morpholin-3-yl]acetamide
3-(3-chlorobenzoyl)-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine
[(1S,3S,3aS,6aR)-3-(5-fluoro-2-methoxyphenyl)-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-6-methyl-4H-pyran-4-one
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(propan-2-ylsulfanyl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(3-fluorophenyl)methyl]-4-[4-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(4-fluorophenyl)piperidin-3-ol
8-(4-hydroxybenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(1R,5S,6R)-3-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-(3-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}-3-oxopropyl)acetamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,4-dimethoxybenzamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(2-methoxy-3-methylbenzoyl)pyrrolidin-3-yl]methanol
1-[(2-chloro-4-fluorophenyl)methyl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(3-{2-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-methyl-N-{1-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
(2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
1-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-yl}morpholine
N-[(4-fluorophenyl)methyl]-3-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}propanamide
2-oxo-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
(3R,9aR)-8-benzoyl-3-benzyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-methylphenyl)methyl]acetamide
1-(3-chlorophenyl)-5-methyl-4-(6-methylpyridine-2-carbonyl)piperazin-2-one
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepane
2-[2-(4-fluorophenyl)ethyl]-4-{4-[2-(thiophen-3-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzene-1,2-diol
1-(cyclopropylmethyl)-N-methyl-5-(quinoline-6-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
2-benzyl-N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide