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(3aS,6aS)-5-(1H-1,3-benzodiazol-2-ylmethyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
2-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}azetidin-3-yl)pyridine
5-(2-fluorophenyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
7-(1,3-benzothiazol-2-yl)-4-(2-methylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3,5-dimethoxyphenyl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
N-[(1S,2R)-2-aminocyclobutyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
1-cyclohexyl-4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepane
N-[(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-ethyl-2-[(3R,4S)-3-methanesulfonamido-4-(4-methoxyphenyl)pyrrolidin-1-yl]acetamide
5-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]pentanoic acid
N'-cyclopentyl-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}butanediamide
5-(isoquinolin-5-yl)pyridine-3-carboxylic acid
N-ethyl-N-(oxan-2-ylmethyl)-1H-1,3-benzodiazole-2-carboxamide
2-fluoro-N-{3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-3-oxopropyl}benzamide
8-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-6-[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-(prop-2-en-1-yl)-N-propyl-1-benzofuran-2-carboxamide
N-[2-(1H-pyrazol-1-yl)ethyl]-4-sulfamoylbenzamide
3-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylaniline
3-methyl-12-(4-phenylphenyl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
4-(2-ethylbutanoyl)-1-phenylpiperazin-2-one
N-methyl-N-[3-(oxolan-2-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-cyclopropylpropanamide
N-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-3-yl)acetamide
6-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}-1H-indazole
[(1R)-1-(3-methoxyphenyl)ethyl]({3-methyl-1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)amine
3-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
5-methyl-3-(1H-pyrazol-3-yl)-2-(4H-1,2,4-triazol-4-yl)pyridine
methyl 7-oxo-9-(3-phenylpropoxy)-3-(quinolin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(3-methoxyphenyl)-1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
3-(3-methoxyphenyl)-1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
1-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(1,3-thiazol-2-yl)piperidine
(3aS,6aS)-2-[(4-methyl-1,3-thiazol-5-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-3-yl)acetamide
1-methyl-8-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(1H-1,2,3-benzotriazol-4-yl)-1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-(2,2-diphenylethyl)-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
4-(2,4-dimethoxyphenyl)-3-[(2-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N,2,6,8-tetramethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
1-[2-(difluoromethoxy)benzoyl]-3-(2,5-dimethoxyphenyl)pyrrolidine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-[(1-ethylpyrrolidin-2-yl)methyl]-15-methyl-13-oxo-9-(thiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[(2-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)hexanamide
N-cycloheptyl-3-(3-propylmorpholin-4-yl)propanamide
N-(4-chloro-2-methoxy-5-methylphenyl)-4-(pyridin-4-yl)piperazine-1-carboxamide