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3-(4-methyl-1H-pyrazol-1-yl)-1-[4-(2-methylphenoxy)piperidin-1-yl]propan-1-one
(1S,5R)-N-[(2-fluorophenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
1-(1-benzofuran-5-carbonyl)-4-(2-methoxyphenoxy)piperidine
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)quinoxaline
4-[(2-methylphenyl)methyl]-3-{2-oxo-2-[4-(piperidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
(4aR,7aS)-1-{2-[methyl(pentyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3aS,6aS)-2-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
8-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
1-(5-acetylpyridin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(1R,3R)-3-aminocyclopentyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
3-propyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
(1S,3R)-N1-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
3-(2-methyl-1H-imidazol-1-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
5-methyl-4-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1-(4-methylphenyl)piperazin-2-one
3-{2-oxo-2-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]quinoline-2-carboxamide
N-(4-fluoro-2-methylphenyl)-3-[1-(3-hydroxypyridine-2-carbonyl)piperidin-3-yl]propanamide
1-benzoyl-2-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidine
N-(2-methyl-1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide
5-(hydroxymethyl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]furan-2-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)benzamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(1-ethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{4-oxo-6-propyl-3H,4H-thieno[2,3-d]pyrimidin-3-yl}propanamide
methyl 3-(2-methoxyacetamido)-1-methyl-5-[(2-methylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}pyrrolidin-3-yl)methyl]benzoic acid
1-(2-methoxyphenyl)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperazin-2-one
4-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)oxane-4-carbonitrile
1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
(4S,4aS,8aR)-1-(4-hydroxy-2-methylpyrimidine-5-carbonyl)-4-phenyl-decahydroquinolin-4-ol
1-methyl-6-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-methoxy-6-[2-(pyrrolidin-1-yl)ethyl]phenyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-3-carboxamide
3-(3-methyl-1H-pyrazol-1-yl)-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
1-cyclopentanecarbonyl-3-(6-methoxynaphthalene-2-carbonyl)piperidine
(1R,5R)-N,N-dimethyl-6-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
N-[3-(azepan-1-yl)propyl]-4-hydroxy-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
2-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}propan-2-ol
3-(2-{[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl]amino}ethyl)-1,3-oxazolidin-2-one
methyl 1-(2-cyclopropyl-1,3-benzoxazole-6-carbonyl)piperidine-2-carboxylate
2-{[6-(8-methylquinolin-5-yl)pyrimidin-4-yl]amino}ethan-1-ol
2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-3-carbonitrile
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-phenylurea
1-(6-chloro-1,3-benzothiazol-2-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}piperidin-4-amine
1-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]piperidin-3-ol