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5-[1-(dimethylamino)propan-2-yl]-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-cyclopropyl-2-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]pyridine-4-carboxamide
2-cyclopentyl-9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3,3-dimethyl-1-({5-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
3-{5-[1-(2-methoxyethyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
3-[3-(piperidine-1-carbonyl)phenyl]-1-{3-[(pyridin-3-yl)amino]propyl}urea
2,6-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
N-(1-phenylethyl)-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N,N-dimethyl-5-{2,4,5-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(17),3,5,7,9,11,13,15-octaen-3-yl}pyrimidin-2-amine
5-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}acetamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1-benzothiophene-5-carboxamide
3-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
2-[(2,3-dihydro-1-benzofuran-2-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(benzylsulfamoyl)({[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl})amine
5-methyl-1'-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({8-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxane-4-carboxamide
N-cyclopentyl-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butanamide
5-fluoro-2-{methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}pyrimidin-4-ol
N-(4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}phenyl)acetamide
3-[4-(3-methoxyphenyl)piperazin-1-yl]-5-phenyl-1,2,4-triazine
N-({7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
2-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-5-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[2-(2-fluorophenyl)ethyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethyl-1H-pyrazole-4-sulfonamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-1-phenylcyclopropane-1-carboxamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(2-oxopyrrolidin-1-yl)benzamide
1-[(2-fluorophenyl)methyl]-N-(2-phenylethyl)piperidin-3-amine
4-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-2-(trifluoromethyl)morpholine
methyl 3-(furan-2-amido)-5-[(4-hydroxybutan-2-yl)amino]-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
[5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)furan-2-yl]methanol
2-[1-(5-chloro-2-methoxyphenyl)-5-(4-cyano-1-methyl-1H-pyrrol-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-{2-[4-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]ethyl}aniline
(1S,4S)-5-(3-hydroxypropanoyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-cyclopentyl-4-methoxy-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzamide
4-[(4aR,8aS)-6-(2-phenylethyl)-decahydro-1,6-naphthyridine-1-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one
4-methanesulfonyl-2-[(4-methoxyphenyl)methyl]morpholine
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-(3-fluoropyridin-2-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-(2-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}-N-[1-(thiophen-2-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-[4-chloro-2-(trifluoromethyl)phenyl]-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
3-ethyl-1-(2-phenylethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-methoxy-4-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-(4-methyl-1H-imidazole-2-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
[(3R,4R)-1-(2,3-dichlorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-{2-[2-(3-fluorophenyl)-6-oxo-1,6-dihydropyrimidin-4-yl]ethyl}acetamide