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2-methyl-4-(5-{[3-(4-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
3-[4-(dimethylamino)phenyl]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
6-chloro-2-[1-(2-ethylpyrimidine-5-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
3-(3-fluorophenoxymethyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 3-benzyl-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidine-3-carboxylate
N-[2-(4-chlorobenzenesulfonamido)ethyl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
2-[(1-cyclohexylpropan-2-yl)amino]-N,N-dimethylethane-1-sulfonamide
3-[6-(dimethylamino)pyridin-3-yl]-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
5-(3-methoxyphenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]furan-2-carboxamide
(1R,5R)-3-(4-chlorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N,5-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-[2-(5-methyl-4-{[2-(trifluoromethyl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)ethyl]-1,4-oxazepane
N-[1-(2-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-3-(2-methoxyphenyl)propanamide
N-[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)methyl]-5-methyl-1,2-oxazole-3-carboxamide
N-(pentan-3-yl)-N-(2-phenylethyl)pyridine-3-carboxamide
3-(cyclohexylsulfamoyl)-5-(1H-pyrazol-3-yl)benzoic acid
6-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-N-propylpyridine-3-carboxamide
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})methylamine
N-cyclohexyl-3-({[(2,2-dimethyloxan-4-yl)methyl]amino}methyl)-N-methylpyridin-2-amine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
methyl 5-{3,7-dioxo-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinolin-9-yl}-2-hydroxybenzoate
N-[2-(2-fluorophenyl)ethyl]-1-(4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N-[7-(4-acetylpiperazine-1-carbonyl)-1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
2-[3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]acetamide
1-[1-(methoxymethyl)cyclobutanecarbonyl]-2-(3-methoxyphenyl)azetidine
(3R,4R)-4-ethyl-1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]piperidine-3,4-diol
3-{2-[4-(4-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
3-[(3R,4S)-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylbenzamide
N-[2-(dimethylsulfamoyl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-ethyl-N-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)acetamide
1-(3-methylphenyl)-N-[2-(morpholin-4-yl)propyl]piperidin-4-amine
methyl 9-[(4-fluorophenyl)methoxy]-3-[(3-hydroxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1H-1,3-benzodiazol-2-ylmethyl)[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]amine
1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}but-2-yn-1-one
N-[(3R,4S)-4-cyclopropyl-1-[2-methyl-2-(piperidin-1-yl)propyl]pyrrolidin-3-yl]-2-hydroxyacetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
1-(carbamoylmethyl)-N-[1-(3-methylphenyl)piperidin-4-yl]piperidine-4-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-3-(trimethyl-1H-pyrazol-1-yl)propanamide
5-(oxolan-3-yl)-4-phenyl-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazole
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methoxy-5-methylbenzoyl)pyrrolidin-3-yl]methanol
7-cyclobutaneamido-N-(furan-2-ylmethyl)-N,1-dimethyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N,N-dimethyl-2-[({thieno[3,2-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-(2,4-dimethylphenyl)-3-{[1-(propan-2-yl)piperidin-4-yl]formamido}propanamide
2-{4-[(6-chloroquinolin-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-cyclohexyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(diethylamino)ethyl]-2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methylacetamide