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(benzylsulfamoyl)({1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl})amine
1,5-dimethyl (2S)-2-{2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]acetamido}pentanedioate
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[2-(4-hydroxyphenyl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
2-(2-{3-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
ethyl 2-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
1-cycloheptyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
4-[(3-hydroxy-3-phenylpropyl)(methyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
6-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
4-methoxy-6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
2-amino-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-4-carboxamide
1-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1H-1,2,3-triazole-4-carboxamide
4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-chloro-N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}thiophene-2-sulfonamide
(3R,4R)-4-methyl-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(propan-2-yl)pyrrolidin-3-ol
2-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,2,3,4-tetrahydroisoquinoline
N-ethyl-N,7-dimethyl-2-[2-(methylamino)pyrimidin-5-yl]quinoline-4-carboxamide
N-[2-(morpholin-4-yl)ethyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-{[1-(2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
1-(4-acetylphenyl)-3-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)urea
N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
6-(4-fluorophenyl)-N-(2-oxopiperidin-3-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4aR,8aR)-4a-hydroxy-7-(6-methoxypyrimidin-4-yl)-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
{4-[(2-chlorophenyl)methyl]-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-4-yl}methanol
(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
methyl 3-(3-ethynylbenzoyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-2-(pyridin-2-yl)acetamide
4-(4-chlorophenyl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]butanamide
3-[2-(4-fluorophenyl)piperidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
4,5,6-trimethyl-2-oxo-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
1-[(3-chlorophenyl)methyl]-4-ethyl-1,4-diazepan-5-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
N,2-dimethyl-5-(propan-2-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
5-methoxy-1-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-indole-2-carboxamide
3-(4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
1-(4-ethylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
N-methyl-2-{3-oxo-2-azaspiro[4.5]decan-2-yl}-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-4-(pyrrolidin-3-yl)benzamide
4-[2-(pyrrolidine-1-sulfonyl)ethyl]-4H-1,2,4-triazole
(4aS,7aR)-1-(5-methylpyrazine-2-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methoxy-1-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-[(2R,3R)-2-hydroxy-1'-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
5-(2-methylphenyl)-2-(pyridin-3-yl)-4-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]pyrimidine
1-(4-{[2-(pyrazin-2-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
N-[1-(methoxymethyl)cyclopentyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
N-[3-(3-methoxyphenyl)phenyl]-1-(2-methylpropyl)piperidine-4-carboxamide