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5-hydroxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyrazine-2-carboxamide
1-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]azetidin-3-ol
benzyl(butyl){[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}amine
3-hydroxy-3-{[(2-methylpropyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
1-cyclohexyl-N3-[(1R)-1-(3-methoxyphenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
(3R,4R)-4-amino-1-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}piperidin-3-ol
methyl 2-[butyl(methyl)sulfamoyl]-6-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[(3-methoxypropyl)amino]-5-methyl-N-[2-(methylsulfanyl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
(3R,5S)-5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-3-ol
N4-methyl-N2-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-4-(5-cyanopyridin-2-yl)piperazine-1-carboxamide
6-fluoro-2-({[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)quinolin-4-ol
N-[3-(2-chlorophenoxy)propyl]-1-ethyl-N-methyl-5-oxopyrrolidine-3-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(4-methylpentan-2-yl)-1,2-oxazole-3-carboxamide
7-methoxy-N,N-dimethyl-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
3-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]pyridin-2-ol
[(3R,5R)-5-(pyrrolidin-1-ylmethyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-yl]methanol
4-(3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanoyl)-1,4-diazepane-1-carbaldehyde
4-{[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)carbamoyl}pyridin-1-ium-1-olate
ethyl 1-{pyrazolo[1,5-a]pyridine-7-amido}piperidine-3-carboxylate
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-{[7-(2-methoxy-2-phenylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
2-(2-methyl-1H-indol-3-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
4-(4-methoxyphenoxy)-1-(oxolan-3-ylmethyl)piperidine
N-[5-(3-acetamidophenyl)-6-methylpyridin-2-yl]propanamide
5-(2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxamide
N,N-dimethyl-2-(4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)acetamide
2-amino-4-(2,3-dimethoxyphenyl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
(1R,2S)-N1-propyl-N2-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]cyclohexane-1,2-dicarboxamide
N-[(3R,4S)-4-cyclopropyl-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}phenol
8-[2-(naphthalen-2-yloxy)propanoyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-[2-(pyridin-2-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(1-ethyl-2-methyl-1H-indol-5-yl)urea
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
6-(cyclopropylmethyl)-3-[(2-methylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-cyclopropyl-4-hydroxy-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrimidine-5-carboxamide
4-[6-(2-methylphenyl)-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyridin-2-yl]morpholine
(2E)-3-(2-chlorophenyl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)prop-2-enamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-(2-fluorophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
6-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-5-[5-(pyridin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-1,2,4-oxadiazole-5-carboxamide
(2S)-2-amino-1-{5-[5-(3-ethyl-1-methyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one
1-[(3-fluorophenyl)methyl]-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
3-[(4-cyclopentylpyrimidin-2-yl)amino]butan-1-ol
2-ethoxy-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}pyridine-3-carboxamide