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2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-fluoro-2-methylphenyl)methyl]acetamide
2-(2-hydroxyethyl)-9-(4-methoxy-3,5-dimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
4-(3-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-2,5-dimethyl-1H-pyrrol-1-yl)-4H-1,2,4-triazole
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
N-cyclopropyl-3-(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
1-ethyl-4-{[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}pyrrolidin-2-one
N-[4-(3-methoxyphenyl)phenyl]-1-(pent-4-enoyl)piperidine-3-carboxamide
6-[(3-methylphenyl)methyl]-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(2-chlorophenyl)-N-{[2-(diethylamino)pyridin-3-yl]methyl}acetamide
4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-1,2-dihydroquinolin-2-one
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[3-(morpholin-4-yl)propyl]amine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
N-(3-methoxyphenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
N-methyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
N-({8-[(2-hydroxy-3-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N-methylpyridine-4-carboxamide
N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-4-(trifluoromethyl)pyrimidin-2-amine
1-pentyl-2-(5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}thiophen-2-yl)pyrrolidine
4-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]azetidin-3-yl}morpholine
4-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-2-[(3-fluorophenyl)methyl]morpholine
N-[(2,3-dimethoxyphenyl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 4-[(3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)methyl]benzoate
methyl 3-[3-(3-methoxyphenyl)propanoyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[2-(dimethylamino)ethyl]-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N,N-diethyl-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-{[4-(methylsulfanyl)phenyl]methyl}-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-cyclopentanecarbonyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
N-[3-(4-chlorophenyl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
N-[2-hydroxy-1-(thian-4-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
6-(2-methoxy-5-methylphenyl)pyridine-3-carboxamide
1-({1-[6-(6-aminopyridin-3-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-phenylpyrimidine-5-carboxamide
7-cyclohexyl-2-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-(5-chloro-2-fluorobenzoyl)-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[(8-methylquinolin-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}morpholin-2-yl)ethan-1-ol
4-hydroxy-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
ethyl 4-{[3-(3-methylpiperidin-1-yl)-3-oxopropyl]amino}piperidine-1-carboxylate
1-(1,3-benzothiazol-2-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}piperidin-4-amine
7-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-(1H-imidazol-1-ylmethyl)piperidine
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
1-ethyl-N,6-dimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2-chloropyridine-4-carbonyl)-N-(3,4-dimethylphenyl)piperidin-3-amine