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[(4-methanesulfonylphenyl)methyl](methyl)[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]amine
3-ethyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxylic acid
2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
3-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)benzoic acid
1-(1-{4-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]phenyl}-2,5-dimethyl-1H-pyrrol-3-yl)ethan-1-one
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(propan-2-yl)propanamide
(2S,4S)-4-amino-N-ethyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
4-(3-fluorophenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
4-cyclobutaneamido-N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)benzamide
5-methyl-3-{3-oxo-3-[2-(pyridin-2-yl)pyrrolidin-1-yl]propyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-{3-methyl-5-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-(propan-2-yl)piperazine
N-methyl-N-{[1-(pyridin-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}cyclohexanecarboxamide
3-(4-methoxyphenyl)-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
2-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
1,3-dimethyl-5-{2-oxo-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl}imidazolidine-2,4-dione
(1S,5R)-6-(2-methyl-1,3-thiazole-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
6-[(diethylamino)methyl]-N-[(1-hydroxycyclohexyl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazole
methyl 3-[(5-methylfuran-2-yl)methyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[5-(5-hydroxypyrazin-2-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-3-(pyridin-3-yl)propanamide
{1-[(2-chlorophenyl)methyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
methyl 3-(furan-2-amido)-6-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
(2E)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(pyridin-3-yl)prop-2-enamide
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[2-(pyridin-4-yl)ethyl]piperidin-4-amine
6-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-methyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
N-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
3,5-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,2-oxazole-4-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1-phenylethyl)benzamide
1-(methoxymethyl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}cyclobutane-1-carboxamide
methyl 6-[2-(3-hydroxyphenyl)-1H-imidazol-1-yl]-1,2,3,4-tetrahydroquinoline-1-carboxylate
8-(2-ethylpyrimidine-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
ethyl 4-{[6-methyl-4-(thiomorpholin-4-yl)quinazolin-2-yl]methyl}piperazine-1-carboxylate
methyl[(4-{2-[4-(4-methylbenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](quinolin-6-ylmethyl)amine
{5-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-ylmethyl]furan-2-yl}methanol
1-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyridin-2-yl)propan-1-one
2-chloro-N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-{1-[1-(but-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
(1S,5R)-3-benzoyl-6-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-fluorophenyl)-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]morpholine
2-{8-[(4-hydroxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide