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(4S,6R)-4-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carbonyl}-6-methyl-1,3-diazinane-2-thione
6-fluoro-2-oxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[2-(dimethylamino)-2-(4-fluorophenyl)-N-(1-methylpiperidin-4-yl)acetamido]acetic acid
1-(4-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-[4-(quinolin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
methyl 7-oxo-3-(pyridin-3-ylmethyl)-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(5-{[3-(5-methylfuran-2-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
6-ethyl-3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
3,6-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-benzofuran-2-carboxamide
(3R,4R)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-[(trimethylpyrazin-2-yl)methyl]piperidin-3-ol
N-[2-(4-chlorobenzenesulfonamido)ethyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
4-[(furan-2-ylmethyl)amino]-N,5-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-benzyl-2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-ethylacetamide
5-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1H-indazol-3-amine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methyl-2-oxopentanamide
3-cyclohexyl-4-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-1H-pyrazole
1-[(2-hydroxy-6-methoxyphenyl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
{1-ethyl-5-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
(1R,2S,9R)-11-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
1-(1H-indazole-3-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
4-(4-methoxyphenoxy)-1-(pyrrolidin-3-ylmethyl)piperidine
2-[benzyl({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]ethan-1-ol
4-[3-(2-phenylethyl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(3-fluorophenyl)methyl]amino}piperidin-1-yl)benzamide
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylbutanamide
3-[(cyclopropylmethyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[2-(cyclohex-1-en-1-yl)ethyl]propanamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
8-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[(2,6-dichlorophenyl)methyl]-5-(4-ethoxypiperidine-1-carbonyl)pyrimidin-4-ol
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(oxan-2-yl)ethyl]acetamide
1-methyl-1'-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-{[2-(1H-indol-3-yl)ethyl]amino}-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-(3-methoxyphenyl)-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propanamide
2-({[(3R,4R)-1-(2-fluoro-6-methoxybenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(diethylamino)-1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(4-fluorophenyl)methyl]-1,2-oxazole-3-carboxamide
ethyl 4-{1-[1-(furan-2-ylmethyl)piperidin-4-yl]piperidin-3-yl}piperazine-1-carboxylate
4-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]pyridine
N-[2-(furan-2-yl)ethyl]-5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-1-(2-methoxyacetyl)-N-methylpiperidine-3-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N,N-bis(prop-2-en-1-yl)benzamide
4-fluoro-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-3-methylthiophene-2-carboxamide
(1R,3S)-7-(5-ethyl-1H-pyrrole-2-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
3-(2-chloro-4-fluorobenzoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide