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3-[(2,4-difluorophenyl)methyl]-N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(furan-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propane-1,2-dione
2-methyl-6-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
4-{4-[methyl(thiophen-3-ylmethyl)amino]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
3-(diethylamino)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-[(4-chlorophenyl)methyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1,2,5-thiadiazole-3-carboxamide
1-(4-fluoro-2-{3-[1-(3-hydroxypropyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
4-{1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]piperidin-3-yl}benzoic acid
(4aR,7aS)-1-(1H-imidazol-2-ylmethyl)-4-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[2-(pyridin-3-yloxy)propyl]pyridin-2-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,2-dimethyl-6-(piperidin-3-yl)pyrimidin-4-amine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-fluorobenzamide
3-{[5-(2-methoxynaphthalen-1-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
N-cyclopropyl-1-{2-[1-(2,3-dimethoxybenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-phenylpentanamide
1-cyclopropyl-5-oxo-N-[(3-phenylphenyl)methyl]pyrrolidine-3-carboxamide
ethyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
7-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4S)-1-[(5-chlorothiophen-2-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
dimethyl(2-{4-[4-(5-methylfuran-2-yl)benzoyl]morpholin-2-yl}ethyl)amine
2-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethoxy}ethan-1-ol
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidine
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(pyrrolidine-1-sulfonyl)benzamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}acetamide
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
(2S)-3-phenyl-2-[(2,3,5,6-tetramethylphenyl)formamido]propanamide
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-(1-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
[(3R,4R)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-(2-methyl-1H-imidazol-1-yl)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidine-4-carboxylic acid
4-[(dimethylamino)methyl]-1-[4-(trifluoromethyl)benzenesulfonyl]azepan-4-ol
N-[(3S)-1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
ethyl 4-(cyclopropylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-methyl-1-(pyrazin-2-ylmethyl)-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
N-({7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
1-phenyl-N-{[1-(thian-4-yl)piperidin-3-yl]methyl}methanesulfonamide
5-[(furan-2-ylmethyl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}benzoic acid
1-{5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-[(3R,4S)-4-(dimethylamino)-1-(3-phenylbenzoyl)piperidin-3-yl]propan-1-ol
(3aR,6aR)-2-cyclopentyl-5-[3-(pyridin-4-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(benzyloxy)methyl]-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
6-{methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one