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N-(oxolan-2-ylmethyl)-3-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]propanamide
2,3-dimethyl-6-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethylbenzamide
4-[(6-methylpyridin-3-yl)oxy]-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidine-4-carboxylic acid
N-[(2-fluorophenyl)methyl]-5-[(1H-indol-2-ylmethyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-ethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(methylsulfanyl)-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-methoxy-N,4-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]benzamide
4-cyclopentyl-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-2-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(3-methylquinoxalin-2-yl)methyl]piperidin-3-amine
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
3-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]propanoic acid
1-(4-ethylpiperazin-1-yl)-3-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenoxy)propan-2-ol
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,4-diazepan-2-one
4-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
4-[(5-chlorothiophen-2-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
methyl 5-(5-chlorothiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N,1-dimethyl-N-[2-(oxan-4-yl)ethyl]piperidin-4-amine
(2S,4R)-4-amino-1-(cyclopentylmethyl)-N,N-diethylpyrrolidine-2-carboxamide
1-cyclopropanecarbonyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3S,4R)-1-(2-ethoxypyridine-3-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
(2R,6S)-2,6-dimethyl-4-[2-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-inden-2-yl]morpholine
2-[4-(6-methyl-2-phenylpyrimidin-4-yl)piperazin-1-yl]propane-1,3-diol
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(4-fluorophenyl)methyl]methylamine
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)propanamide
1-(azepan-1-yl)-2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
1-{4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-cyclobutanecarbonyl-N-(2-ethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
(3aR,6aS)-N-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
N-(cyclopropylmethyl)-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
1-{4-[(3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}ethan-1-one
methyl (2S,4R)-4-[4-(azepan-1-yl)-4-oxobutanamido]-1-methylpyrrolidine-2-carboxylate
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
2-amino-6-(4-hydroxyphenyl)-4-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]pyridine-3-carbonitrile
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
N-cyclopropyl-4-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperazine-2-carboxamide
N-(3-fluorophenyl)-6-(2-methylbutyl)-6-azaspiro[2.5]octane-1-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
(2R)-N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]oxolane-2-carboxamide
N-{[7-(9-methyl-9H-carbazole-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
2-methyl-6-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]pyrimidin-4-ol
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(furan-3-ylmethyl)methylamine
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methylthiophene-2-carboxamide