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[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl]methylamine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[2-(4-chlorophenyl)-2-hydroxyacetyl]piperazin-1-yl}-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-ethyl-1-(propan-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-(2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}ethyl)-N-methylmethanesulfonamide
2-methyl-6-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
N-[(4,5-dimethylfuran-2-yl)methyl]-1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-(1-cyclopentanecarbonylpiperidin-4-yl)-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-[(furan-2-ylmethyl)amino]-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-(dimethyl-1,2-oxazol-4-yl)-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-{[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]amino}pyridine-3-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(pyridin-2-yl)ethyl]benzamide
5-ethyl-2-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
3-(cyclopropylmethyl)-1-(2-methoxyethyl)piperidine-3-carboxylic acid
(2R)-2-amino-3-(ethylsulfanyl)-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
2-(2,4-difluorophenoxy)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
methyl 4-({2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamido}methyl)benzoate
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(4-hydroxy-3-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-amine
2-cyclopropyl-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-methyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(2S,4S)-4-amino-1-[3-methyl-4-(morpholin-4-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-[(2-methoxyethyl)(methyl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-(2-phenylethyl)acetamide
N-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methyl]-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(methoxymethyl)-N-[(4-sulfamoylphenyl)methyl]thiophene-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-[(methylsulfanyl)methyl]-N-(4-phenoxyphenyl)piperidine-1-carboxamide
1-(5-methylthiophene-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
6-[(diethylamino)methyl]-N-(1-methyl-6-oxopiperidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
3-{2-[4-(2-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-1-ethyl-3-(2-methylphenyl)pyrrolidine-2,5-dione
N-{2-[3-(3-methylbutoxy)phenyl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
N-(2-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
2-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-5-methoxy-1-methyl-1H-indole
dimethyl[2-(2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
4-(5-methoxy-1H-indole-2-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
6-[(3-methoxyphenyl)methoxy]-4-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
2-methyl-9-(6-methylpyridine-2-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
2-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)benzonitrile
2-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1-methylazepane