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(2R,6R)-1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-(1-cyclohexylpiperidin-3-yl)-4-phenylpiperazine
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-(1H-pyrazol-5-yl)piperidine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
7-[(3-methylphenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentyl-4-(1H-1,2,3-triazole-5-carbonyl)-1,4-diazepane-6-carboxylic acid
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[4-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-methoxypyridine-4-carboxamide
1-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]cyclopentane-1-carbonitrile
1-(morpholin-4-yl)-3-{5-[2-(oxolan-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-{[4-(2-cyclobutylacetyl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzoic acid
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[4-(1H-imidazol-1-yl)phenyl]urea
(2R,3S,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
{3-[(3-chlorophenyl)methyl]-1-(4-fluorobenzenesulfonyl)piperidin-3-yl}methanol
4-[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-methylpiperidine
N-[(3,5-difluorophenyl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
3-(4-chlorophenyl)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-propyl-4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
1-benzyl-3-(pyridin-2-ylmethyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-(trifluoromethyl)pyrimidin-2-amine
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(5-propyl-1,2-oxazol-3-yl)formamido]methyl}benzoate
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
5-cyclopropanecarbonyl-1'-(2-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-cyclopentyl-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-2-one
methyl 5-[(7-methyl-1H-indol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(1S,5R)-N-(3-methoxyphenyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}morpholine
(2S,4S)-4-amino-1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxylic acid
(5S,9aS,9bS)-2-cyclopentyl-5-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(pyrrolidin-2-yl)-N-(1H-1,2,4-triazol-5-ylmethyl)thiophene-2-carboxamide
(3aR,7aS)-2-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-(1H-imidazol-2-ylmethyl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenoxy)piperidine
4,6-dimethyl-3-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]-1,2-dihydropyridin-2-one
4-[(2-chlorophenyl)methyl]-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-{[4-(aminomethyl)phenyl]methyl}-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(1-methyl-1H-pyrrole-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2,4-dimethoxybenzoyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine
(1R,5R)-6-benzyl-3-cyclopropanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
methyl 3-(4-fluorobenzenesulfonamido)-5-{[2-(thiophen-3-yl)acetamido]methyl}benzoate
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-[2-(difluoromethoxy)phenyl]pyridine-3-carbonitrile
4,6-dimethyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-cyclopentanecarbonyl-3-(2-methoxybenzoyl)piperidine
methyl 8-(1-benzothiophen-2-ylmethyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate