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1-(2-{5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}ethyl)pyrrolidin-2-one
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-1-(2-methoxyethyl)pyrrolidine-3-carboxamide
4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(2-phenylethyl)morpholine
3-[(3R,4S)-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N,N-diethyl-6-fluoro-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
3-chloro-4-fluoro-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzothiophene-2-carboxamide
ethyl 4-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)piperidine-1-carboxylate
(3S,5R)-N3-[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
(2S)-3-methyl-2-({[3-(sulfamoylmethyl)phenyl]carbamoyl}amino)butanamide
1-[4-({3H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(5-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-[4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-2-(cyclopent-1-en-1-yl)ethan-1-one
3-(3-hydroxy-3-methylbutyl)-N-[(3-methoxyphenyl)methyl]benzamide
N-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-2-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(3-ethoxypropyl)amine
(2S,4S)-4-amino-N-methyl-1-[3-(4-methylbenzenesulfonyl)propanoyl]pyrrolidine-2-carboxamide
4-[(3-fluoro-4-methylphenyl)methyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-4-sulfamoylbenzamide
2-(cyclohex-1-en-1-ylmethyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 4-(methylsulfanyl)-2-({6-phenylimidazo[2,1-b][1,3]thiazol-3-yl}formamido)butanoate
[1-(4-aminopyrimidin-2-yl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
3-(furan-2-yl)-1-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
N-{[1-(1,3-benzothiazole-6-carbonyl)-4-hydroxyazepan-4-yl]methyl}methanesulfonamide
1-(2-cyclohexylethyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(methylcarbamoyl)cyclohexyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
(2S)-2-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-4-(methylsulfanyl)butan-1-ol
2-benzyl-8-(2-phenoxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(4-methylpiperidin-1-yl)pyridine-3-carboxamide
6-benzyl-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-(2-{4-[(2-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methoxy-1-{4-methyl-2-[3-(3-methylphenoxy)azetidine-1-carbonyl]piperazin-1-yl}ethan-1-one
N-[2-(1H-imidazol-1-yl)ethyl]-5-[1-(3-methylbutyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-methylacetamide
1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
1-(benzyloxy)-8-(3-methylfuran-2-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
5-oxo-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidine-3-carboxylic acid
3-chloro-4-fluoro-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]propanamide
1-(1H-imidazol-2-ylmethyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(pyrazin-2-yl)propan-1-one
N-(cyclopropylmethyl)-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-propylpropanamide
N-ethyl-2-[4-(2-methoxypyridine-4-carbonyl)piperazin-1-yl]acetamide
3-{1-[(3-chloro-4,5-dimethoxyphenyl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
N,N,2-trimethyl-7-(7-methyl-1-benzofuran-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(2-chloro-4-fluorophenyl)methyl]piperazin-2-one
ethyl 4-[1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
N-[2-(2,5-dimethylphenoxy)ethyl]-5-(methoxymethyl)-N-methylfuran-2-carboxamide
4-(4-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}phenyl)-2-methylbutan-2-ol
4-(4-hydroxy-3-methylbenzoyl)-1-(2-methylphenyl)piperazin-2-one