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N-(2-fluoroethyl)-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)sulfonyl]benzamide
methyl (3aS,6aS)-2-(6-methylpyridine-2-carbonyl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
(3R,4R)-1-(4-chloro-2-fluorobenzoyl)-4-cyclobutyl-3-methylpiperidin-4-ol
(1R,9aR)-1-({[3-(2-ethyl-1H-imidazol-1-yl)propyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}(1-methoxypropan-2-yl)amine
4-[2-(furan-2-yl)phenyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]acetamide
3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1-[3-(trifluoromethyl)phenyl]urea
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-4-methylpyrimidine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1,3-benzothiazole-6-carboxamide
1-{1'-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-[(propan-2-yl)amino]-N-[1-(thian-4-yl)piperidin-4-yl]pyrimidine-5-carboxamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
N3-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-N1-(5-methylpyridin-2-yl)propane-1,3-diamine
5-(3,3-dimethylbutanoyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-ethyl-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4-methyl-1H-pyrazole-5-carboxamide
4-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propane-1,3-diol
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(2-aminoethyl)-N-[2-(propan-2-yloxy)ethyl]quinazolin-4-amine
1-(2-methoxyethyl)-5-(5-methylthiophene-2-carbonyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-acetamido-1-(2-methoxyethyl)-N-[3-(methylsulfanyl)propyl]-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
1-(carbamoylmethyl)-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]piperidine-3-carboxamide
(3aS,6aR)-5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(oxolan-2-ylmethyl)acetamide
4-(1-hydroxyethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
(5S)-5-{[(pyridin-4-ylmethyl)({[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyrrolidin-2-one
1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
methyl 1-[3-(2H-1,3-benzodioxol-4-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
N-[1-(3,5-difluorophenyl)cyclopropyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 2-{8-[(2-hydroxy-3-methoxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
4-{2,2-dimethyl-3-[4-(3-methylpyridin-4-yl)piperazin-1-yl]propyl}morpholine
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}acetamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
1-methyl-4-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,4,9-triazaspiro[5.5]undecane
6-cyclopentyl-N,1-dimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-(4-{[(4-phenyloxan-4-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
5-(2,4-difluorophenoxymethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
N-(1-hydroxy-2-methylpropan-2-yl)-2-[2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]acetamide
2-(4-fluoro-2-methylphenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
4-(1-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)morpholine
N-propyl-N-(pyridin-3-ylmethyl)-3-(pyrimidin-2-yloxy)benzamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
2-[(1-cyclopentylpiperidin-2-yl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one