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5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
N-(3-methoxypropyl)-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}propanamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]propan-1-one
(1S,5R)-6-[(2,6-dichloro-3,4-dimethoxyphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-({2-[1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
5-methyl-3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-(2,3-dimethoxyphenyl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-imidazole
methyl 3-{[1-(cyclopropylmethyl)-5-[4-(pyrrolidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxypyridine-3-carboxamide
(1S)-1-(3-cyclopentyl-1-ethyl-1H-1,2,4-triazol-5-yl)-2-phenylethan-1-ol
3-methyl-N-(2-oxoazepan-3-yl)-5-(phenoxymethyl)furan-2-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
N-(2-methylphenyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
(3R,4R)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dimethylpyrrolidin-3-ol
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
5-methyl-3-(thiophen-3-ylmethyl)-5-{1-[(2,4,6-trimethoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(5-acetylthiophen-3-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
4-(cyclohex-3-en-1-yl)-1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1H-1,2,3-triazole
N-[(2,6-difluorophenyl)methyl]-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(piperidin-1-yl)propan-1-one
4-(1-benzofuran-2-yl)-2-[4-(4-ethylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]pyrimidine
N-({1-[2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}methyl)acetamide
1-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(1S,5R)-6-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-benzyl-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
8-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-benzothiophene-2-carboxamide
5-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidine
5-[4-(2-methoxyethoxy)piperidine-1-carbonyl]-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
4-(1H-imidazol-2-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidine
3-[1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-N-(2-phenylethyl)formamido]propanamide
4-[2-(2,3-dimethylphenoxy)acetyl]-1-[(2-fluorophenyl)methyl]piperazin-2-one
2-amino-3-ethyl-N-[(1-phenylcyclopentyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-{2-[(4aS,8aR)-decahydroisoquinolin-2-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-cyclopropyl-N-methyl-6-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-(thiophen-2-ylmethyl)benzamide
5-[1-(dimethyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(2-phenylethyl)-7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl](2-phenylpropyl)amine
1-methyl-N-(pyridin-4-ylmethyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-amine
6-(4-ethyl-5-methylpyrimidin-2-yl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[(4-hydroxyphenyl)methyl]piperidine-3-carboxylate
2-(2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethoxy)ethan-1-ol
2-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one