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3-(1H-1,3-benzodiazol-2-yl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[3-(3,4-dimethylphenoxy)propyl]-N,4-dimethyl-2-(methylamino)-1,3-thiazole-5-carboxamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-2-yl)methyl]acetamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)propanamide
2-methyl-8-{[3-(5-methylfuran-2-yl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine
3-(hydroxymethyl)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidin-3-ol
5-benzenesulfonamido-N-(2,2-dimethyloxan-4-yl)-1-ethyl-2-methyl-1H-1,3-benzodiazole-7-carboxamide
3-methoxy-5-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}thiophene-2-carboxamide
4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)morpholine
2-{9-[(4-chloro-3-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
3-(furan-2-yl)-1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)propan-1-one
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
2-[2-(2-methyl-1,4-oxazepan-4-yl)-2-oxoethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-[1-(hydroxymethyl)-9-(2-phenylethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(methylsulfanyl)ethan-1-one
6-[4-(1-ethoxyethyl)phenyl]pyrazine-2-carboxylic acid
3-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
5-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
9-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
14-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(4aR,8aS)-6-[(2E)-3-phenylprop-2-en-1-yl]-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2-(cyclopropylmethyl)-8-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(6-phenoxypyridin-3-yl)-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxamide
3-[(1-acetylpiperidin-4-yl)oxy]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-4-methoxybenzamide
2-amino-6-(4-chlorophenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
4-[4-(3-methylpiperidine-1-carbonyl)phenoxy]-1-(2-phenylethyl)piperidine
N-{2-[1-(quinolin-4-ylmethyl)piperidin-3-yl]ethyl}methanesulfonamide
1-(4-fluorophenyl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
2-[2-(4,5,6,7-tetramethyl-1H-1,3-benzodiazol-2-yl)phenoxy]acetamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4-methyl-3-oxopiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-{1-[2-(naphthalen-2-yl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
8-(butan-2-yl)-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-methoxyphenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
N-(oxolan-3-yl)-2,2-diphenylacetamide
4-[(2-methoxypyrimidin-5-yl)methyl]-3-propylmorpholine
1-(2-methoxyphenyl)-N-[1-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-4-chloro-1-methyl-1H-pyrazole-3-carboxamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[(2-methoxyphenyl)methyl]propanamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
(3S,4R)-4-(3-methoxyphenyl)-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
1-cyclobutanecarbonyl-N-[2-(2-methyl-1H-indol-3-yl)ethyl]piperidine-4-carboxamide
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-(2-{1-[2-(2,5-dimethylphenyl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-cyclobutyl-N-methyl-N-(2-phenylethyl)piperidin-3-amine
5-(2-chloro-6-fluoro-3-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-[2-(2-fluorophenyl)ethyl]-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
N-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-6-methoxy-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-methyl-N-[(2-methylphenyl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide