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[1-(1H-imidazol-1-yl)propan-2-yl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidine-2-carboxamide
2-cyclopropyl-9-[3-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4'-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-benzyl-N-(cyclobutylmethyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
6-ethyl-2-methyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}quinoline-4-carboxamide
4-{[4-(2-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-2-yl}ethoxy)phenyl]methyl}piperazine-1-carbaldehyde
3-{1-[(4,4-dimethylpiperidin-1-yl)sulfonyl]piperidin-3-yl}benzoic acid
2-ethoxy-6-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenol
N-benzyl-2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}acetamide
2-(2-{methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-(pyridin-2-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
5-[2-(methylsulfanyl)acetyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(2,2-diphenylethyl)-4-(1H-pyrazole-4-carbonyl)morpholine
4-(6-hydroxy-1,4-oxazepan-4-yl)-2-methoxypyridine-3-carbonitrile
6-(4-{[3-(dimethyl-1,2-oxazol-4-yl)propyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
8-[(4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-3-ylmethyl)piperazine-1-carboxamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(cyclohexylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-hydroxycyclohexyl)methyl]acetamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}propanamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3-methylcinnolin-5-yl)-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-(methylamino)acetamide
5-acetyl-2,4-dimethyl-N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]-1H-pyrrole-3-carboxamide
1-(2-phenylethyl)-8-(propan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[2-(4-fluorophenyl)acetamido]methyl}benzoate
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
9-methoxy-10-(thiomorpholine-4-carbonyl)-3-(2,4,5-trifluorobenzoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
3-ethyl-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
4-(2,6-dimethoxybenzoyl)-7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}[1-(1H-imidazol-1-yl)propan-2-yl]amine
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
(1S,5R)-6-[(2-fluoro-4-methoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(trifluoromethyl)benzamide
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-{[2-(methoxymethyl)piperidin-1-yl]methyl}benzoic acid
(4aR,7aS)-1-[2-({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3-{[1-(2-cyclopropylquinoline-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](furan-3-ylmethyl)methylamine
1-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(prop-2-en-1-yl)urea
2-(3-methyl-1H-pyrazol-1-yl)-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-{3-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]propyl}pyrrolidin-2-one
4-(azonan-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]pyridine-2-carboxamide
3-(2-chlorophenyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
diphenyl(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methanol
N'-(3-chloro-2-methylphenyl)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanediamide