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6-(2,5-dimethoxyphenyl)-N-methyl-2-(4-methylpiperazin-1-yl)-N-(1-methylpiperidin-4-yl)pyridine-3-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-ethyl-1-methyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-1H-pyrazole-5-carboxamide
1-(2-methoxy-4-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[2-(pyridin-4-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
3-[1-(2,4-dimethyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-3-yl]benzoic acid
1-(piperidin-3-ylmethyl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(butan-2-yl)-2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
3-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-2-yl}pyridine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-[6-(methoxymethyl)pyrimidin-4-yl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
5-(4-benzylpiperidine-1-carbonyl)-1-cycloheptylpiperidin-2-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyridin-2-yl)piperazine
7-(4-fluoro-2-methylbenzenesulfonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
N3-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
N-methyl-N-[(4-phenoxyphenyl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
5-butyl-1'-(1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
4-({2-[1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-{[(benzylsulfamoyl)amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1H-pyrazole-4-carboxamide
2-tert-butyl-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyrimidin-4-ol
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl][(4-fluoro-3-methoxyphenyl)methyl]amine
1-{4-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
N-cyclopropyl-N-[(4-ethylphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
4-(5-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)morpholine
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(4-methylpiperazin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-{[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenol
N,5-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-phenyl-1,2-oxazole-4-carboxamide
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-(2-phenylethyl)piperazine
N-(3-hydroxy-3-phenylpropyl)-N-methyl-3-(2-oxopiperidin-1-yl)propanamide
N-methyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,6-dimethoxypyridine-3-carboxamide
4-(3-chloropyridin-4-yl)-1-[(3-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-benzyl-8-[(2-chloro-6-fluorophenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[3-(1H-imidazol-1-yl)propyl]amino}-N-[1-(4-methylphenyl)ethyl]acetamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
6-chloro-2-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)quinoline
1-{1-[3-(difluoromethoxy)benzoyl]piperidin-3-yl}-2-phenylethan-1-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]acetamide
2-{4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperazin-1-yl}-N-(propan-2-yl)acetamide
1-cycloheptyl-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
3-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one