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4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-(oxolan-3-ylmethyl)piperidine
10-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
1-(2-phenylethyl)-N-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[3-(propan-2-yloxy)propyl]acetamide
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
7-(propan-2-yl)-2-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-(cyclohexylmethyl)-3-hydroxy-3-[(4-methylpiperidin-1-yl)methyl]piperidin-2-one
(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(oxan-2-ylmethyl)piperidin-4-yl)methanol
6-methoxy-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrimidin-4-amine
N-(2,4-dimethoxyphenyl)-3-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)propanamide
2-methyl-N-{2-oxo-2-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}propanamide
2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-8-fluoroquinolin-4-ol
2-(3-hydroxypropyl)-9-(5-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
1-(cyclopropylmethyl)-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2-methoxyphenyl)acetamide
7-methyl-2-[4-(pyrimidin-2-yloxy)phenyl]-1H-1,3-benzodiazole
7-[2-(4-fluorophenyl)morpholine-4-carbonyl]quinolin-8-ol
2-(3-methoxyphenoxy)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
5-fluoro-2-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
[(1-benzyl-1H-pyrazol-4-yl)methyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
5-(2-chlorophenyl)-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]furan-2-carboxamide
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[2-(methylsulfanyl)benzoyl]piperidine
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-chlorobenzamide
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
(1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)methanol
[(3,5-difluorophenyl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-phenyl-5-[1-(pyrazin-2-yl)propan-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-chloro-2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
1-{[3-(difluoromethoxy)phenyl]methyl}-3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)urea
2-(cyclopropylmethyl)-9-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(2,3-difluorophenyl)methyl]-2-(4-methoxybenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
1-[6-(3-methyl-1H-pyrazol-5-yl)pyridazin-3-yl]azepane
3-[4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
{1-[(3,5-dichloropyridin-4-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
6-(cyclopropylmethoxy)-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-{1-[(2-methylphenyl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
7-[(3,4-difluorophenyl)methyl]-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
3-cyclopropyl-5-[(E)-2-phenylethenyl]-1H-1,2,4-triazole
4-(3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]ethan-1-one
1-(2,6-dimethoxypyridin-3-yl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea