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1-phenyl-4-[4-(pyrrolidin-1-ylmethyl)benzoyl]-1,4-diazepane
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
2-(2-aminoethyl)-N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)quinazolin-4-amine
4-(3-{[(benzyloxy)carbonyl]amino}pyrrolidine-1-carbonyl)benzoic acid
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-ethylpyrimidine-5-carboxamide
4-chloro-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
1-methyl-4-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}sulfonyl)piperazine
methyl 6-[(3aS,6aR)-2-oxo-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-3-carboxylate
3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
1-benzyl-6-(pyridin-2-ylmethoxy)-4-[2-(pyridin-2-ylsulfanyl)acetyl]-1,4-diazepan-2-one
N-propyl-N-(pyridin-3-ylmethyl)adamantane-1-carboxamide
9-{5-[(dimethylamino)methyl]furan-2-carbonyl}-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinoline-4-carbonyl)piperidin-3-yl]propan-1-ol
5-{2-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})[1-(pyridin-4-yl)ethyl]amine
N-{2-[2-(phenylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
1-(cyclopropylmethyl)-6-(furan-3-carbonyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N4-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
(2S,4R)-4-amino-N-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
2-(5-fluoro-2-methoxyphenyl)-6-methylpyridine-3-carboxylic acid
(4aS,7aR)-1-(1H-indole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{2-azabicyclo[2.2.1]heptane-2-carbonyl}piperidin-1-yl)-4,6-dimethylquinazoline
N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
2-amino-6-cyclopropyl-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
3-methyl-N-[3-(5-methyl-4-{[3-(4-methyl-1,3-thiazol-5-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]butanamide
3-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2,3-dimethoxybenzamide
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(1-phenylcyclopropyl)propanamide
3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-2,6-dimethylquinoline
9-(1H-1,2,3-benzotriazole-5-carbonyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(pyrazin-2-yl)ethyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
4-[(1E)-3-[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]prop-1-en-1-yl]-2-methoxyphenol
N-({4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)quinoline-2-carboxamide
(3aR,6aS)-5-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclopentyl-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-1,4-diazepane
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-(propan-2-yl)pyrimidin-4-amine
4-{2-[4-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]ethyl}morpholine
(1R,5R)-6-(cyclohexylmethyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-2-(methylamino)pyridine-4-carboxamide
(3R,4R)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(2H-1,3-benzodioxol-5-yl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-[(2,6-dichlorophenyl)methyl]-N-ethyl-4-hydroxy-N-(2-hydroxyethyl)pyrimidine-5-carboxamide
N-(butan-2-yl)-4-(5-{[(3-fluorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidine-1-carboxamide
N-benzyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-ethoxy-3-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine