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4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(3-methylpyridin-4-yl)methyl]benzamide
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-[(1H-1,2,3,4-tetrazol-5-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
N-(2-methylphenyl)-N'-{[1-(morpholin-4-yl)cycloheptyl]methyl}propanediamide
3-(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
1-{7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
ethyl 1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-4-(cyclopropylmethyl)piperidine-4-carboxylate
2-(2-{[3-(1H-imidazol-1-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[(1-benzylpiperidin-4-yl)methyl]-2-(1-cyclopentyl-3-oxopiperazin-2-yl)acetamide
1-methyl-2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-{2-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-3-methoxypropanamide
3-cyclohexyl-1-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propan-1-one
(3S,4S)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
methyl 3-(3,5-dimethylbenzoyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)pyrrolidine-2,5-dione
8-[6-(dimethylamino)pyrimidin-4-yl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
6-(2-chlorophenyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{3-[4-(2-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-ethyl-2-[4-(3-methoxybenzoyl)piperazin-1-yl]pyridine-3-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-methoxy-1-(4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-(1-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
methyl 5-{[(2-fluoro-5-methoxyphenyl)methyl]amino}-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyridazine
3-(2,5-difluorobenzoyl)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]piperidine-3-carboxamide
6-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}benzamide
[(5-ethylpyridin-2-yl)methyl]({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
N4-[(5-methylpyrazin-2-yl)methyl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
7-[cyclohexyl(methoxy)methyl]-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
N-(4-acetylphenyl)-3-oxa-9-azaspiro[5.5]undecane-9-carboxamide
2-{[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzonitrile
methyl 3-({cyclopropyl[(3-hydroxyphenyl)methyl]carbamoyl}amino)-4-methylbenzoate
N-(2H-1,3-benzodioxol-5-yl)-1-(5-chlorothiophene-2-carbonyl)piperidin-3-amine
[(3S,4S)-1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(hydroxymethyl)pyrrolidin-3-yl]methanol
2-ethyl-1-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}butan-1-one
1-cycloheptanecarbonyl-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(1-methylpiperidin-3-yl)ethyl]propanamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
ethyl 1-(2,4-dimethylphenyl)-5-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-1H-pyrazole-4-carboxylate
2-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine
1-(4-methoxyphenyl)-2,2-dimethyl-4-(4-methyl-1,3-thiazol-2-yl)piperazine
N-{[8-(9H-fluoren-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-methoxyacetamide
5-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
2-(ethylsulfanyl)-1-{1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one