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3-[2-(ethylsulfanyl)ethyl]-1-[1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
7-(1-methyl-1H-indole-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N4-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
2-methyl-1-{4-[(3S,4R)-3-(propan-2-yl)-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]piperidin-1-yl}propan-1-one
{3-cyclobutanecarbonyl-9-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(3aR,6aS)-5-(3-cyano-5-fluorobenzoyl)-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N2,N2,N4-trimethyl-N4-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
4-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
N-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-(morpholine-4-carbonyl)piperidin-4-amine
2-(4-{[(furan-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-(piperidin-3-yl)-3,4-dihydropyrimidin-4-one
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(6-methylpyridine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-chloro-N-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-cyclobutyl-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
6-[(4-fluorophenyl)methoxy]-4-[2-(1H-imidazol-2-yl)benzoyl]-1-(propan-2-yl)-1,4-diazepan-2-one
2-{2-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]propyl}pyrazine
2-(4-chloro-2-{[4-(dimethylcarbamoyl)piperazin-1-yl]methyl}phenoxy)acetic acid
6-{2,7-diazaspiro[4.5]decane-2-sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}ethan-1-one
2-(5-methyl-1H-pyrazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
(3S)-1,3-dimethyl-4-(2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
1-(1H-imidazol-2-ylmethyl)-4-(2-methoxybenzoyl)piperazine
3-(2-methoxyphenoxy)-1-(3-methylfuran-2-carbonyl)azetidine
2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(thiophen-3-yl)acetic acid
2-[(3,5-difluorophenyl)methyl]-8-(pyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-2-(4-fluorophenyl)ethyl}-N-methyl-3-(methylsulfanyl)propanamide
2-{methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}acetic acid
N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
4-acetyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
[(3S,5R)-1-(5-ethyl-1,2-oxazole-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-[(2,4-dimethoxyphenyl)methyl]-4-{4-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
1-[5-methoxy-2-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-(oxan-2-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-1-(2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-oxoethyl)-1H-indole-3-carbonitrile
2-(dimethylamino)-2-(4-methylphenyl)-N-[1-(thian-4-yl)piperidin-4-yl]acetamide
2-{1-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}quinoline-2-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-chloro-6-methoxy-4-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}phenol
4-[1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-ethylphenyl)methyl]-N-methylacetamide
N-butyl-N-(4-hydroxybutyl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
6-[1-(3,5-dichloro-4-methylbenzoyl)piperidin-3-yl]pyrimidin-4-ol
(9aR)-N-benzyl-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-[2-(3-chlorophenyl)ethyl]-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide