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8-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyridin-2-yl)piperazine-1-carbonyl]quinoline
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-phenyl-1H-1,2,3,4-tetrazol-5-amine
2-methyl-6-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-phenylpyrrolidine-2,5-dione
2-cyclopropanecarbonyl-8-(5-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2-methoxy-4-methylphenoxymethyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
3-methyl-N-{2-[methyl(phenyl)amino]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
N,N-dimethyl-5-(3-{1-[(3-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)furan-2-carboxamide
3-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazole
1-(2-phenylpropyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-methyl-3-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-fluoro-N-{3-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}benzamide
8-[(3,5-dimethoxyphenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
2-{4-[4-(propan-2-yl)pyrimidin-2-yl]morpholin-2-yl}ethan-1-amine
methyl 3-acetamido-5-[(4-methoxy-4-methylpentan-2-yl)amino]-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl (2S,4S)-4-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetamido]-1-methylpyrrolidine-2-carboxylate
8-[(4-fluoro-2-methylphenyl)methyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-methoxyphenyl)-2-{2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
2-{4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)(methyl)amino]ethan-1-ol
methyl 5-{[(2-chlorophenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(3-phenylbenzoyl)pyrrolidin-3-yl]methanol
N-(1-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
5-{[(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-[2-(thiophen-2-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-amino-N-ethyl-1-[2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetyl]pyrrolidine-2-carboxamide
(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
(3S,4R)-1-[2-(methylsulfanyl)benzoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(2S,4R)-N-[2-(dimethylamino)ethyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
(1H-imidazol-4-ylmethyl)({[4-(methylsulfanyl)phenyl]methyl})propylamine
4-(azepane-1-carbonyl)-6,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
N-{2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}ethane-1-sulfonamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]acetamide
{3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]phenyl}methanol
9-[2-methyl-5-(trifluoromethyl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-[5-(2-ethylbutyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-methyl-1,2-dihydroquinolin-2-one
3-[(2-methoxyphenyl)methyl]-3H,4H-pyrido[2,3-d]pyrimidin-4-one
4-(3,4-difluorobenzoyl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
1-[3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenoxy)propyl]-4-methylpiperazine
1-(1-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1H-indol-3-yl)ethan-1-one
3-chloro-5-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
(4aR,7aS)-1-ethyl-4-(6-phenylpyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(3,4-dimethoxyphenyl)-4-(furan-3-ylmethyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4R)-4-amino-1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide