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N-[(2R,3R)-2-methoxy-1'-[(2,3,6-trifluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
(1-{[1-(2-fluorobenzenesulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
6-(2-aminoethyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methylpyrimidin-4-amine
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-(phenylcarbamoyl)piperidine-3-carboxylate
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
methyl 3-{4-[4-methyl-2,5-dioxo-1-(thiophen-3-ylmethyl)imidazolidin-4-yl]piperidine-1-carbonyl}benzoate
N-cyclopropyl-1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}piperazine-2-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[(5-methylpyrazin-2-yl)methyl]urea
N-{3-[4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]phenyl}pyridine-3-carboxamide
4-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
2-(4,5-dichloro-1H-imidazol-1-yl)-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
3-methyl-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]but-2-en-1-one
N-[(4-methoxyphenyl)methyl]-1-(2-methyloxane-2-carbonyl)piperidine-4-carboxamide
4-{5-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
(3aR,6aR)-2-(2-hydroxyethyl)-5-[(5-phenylthiophen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N'-benzyl-N-(3,5-dimethylphenyl)propanediamide
2-{9-[(3-ethylphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-[3-(4-fluorophenoxy)propyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
ethyl 4-methyl-3-(2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamido)pentanoate
N-(2-methylpropyl)-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-6-[(1-methyl-1H-imidazol-5-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(3-cyanophenyl)-3-({methyl[2-(methylcarbamoyl)ethyl]amino}methyl)benzamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-[3-(1H-imidazol-1-yl)propyl]-1-methylpyrrolidine-3-carboxamide
(3S,4R)-1-[(5-ethylpyridin-2-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
6-[4-(furan-2-yl)benzoyl]-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
(3R,9aR)-3-benzyl-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-[(3-methoxyphenyl)methyl]-2-propanoyl-2,7-diazaspiro[4.5]decan-6-one
4-{5-[1-(3-fluoropyridine-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
1-{1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-[4-(2,3-dimethylphenyl)piperazin-1-yl]ethan-1-one
N-[(2,3-dimethoxyphenyl)methyl]-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
3-[4-(aminomethyl)phenyl]-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
3-[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
1-(4-methoxyphenyl)-4-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}butane-1,4-dione
3-(2-methoxy-5-phenylphenyl)-1-methyl-1-(oxan-2-ylmethyl)urea
N-cyclopentyl-3-{[2-(pyrrolidin-1-yl)ethyl]sulfamoyl}benzamide
2-[(3S,4R)-3-cyclopropyl-4-[2-(pyridin-3-yl)acetamido]pyrrolidin-1-yl]-N-methylacetamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(thiophen-3-yl)ethan-1-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(4-phenyl-1,3-thiazol-2-yl)methyl](pyridin-4-ylmethyl)amine
3-(3-methoxy-6-methylpyridin-2-yl)quinoline
(1S,5R)-3-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[(2,3-difluorophenyl)methyl]-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R)-3-(1,4-oxazepan-4-yl)-1'-(pyrazin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl 6-[(2-ethoxyphenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide