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N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethan-1-one
3-(hydroxymethyl)-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidin-3-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)but-3-enamide
methyl 6-{2-[(2,2-dimethylpropanamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}pyridine-3-carboxylate
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-(2,3-difluorophenyl)-N-methylacetamide
1-[(dimethyl-1,3-thiazol-5-yl)methyl]-5,5-diphenylpiperidin-2-one
1-[(3-methoxyphenyl)methyl]-N3-methyl-N5-[(4-methylphenyl)methyl]-4-oxo-N3-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[(4-methylphenyl)methyl]acetamide
3-ethyl-1-methyl-4-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}piperazin-2-one
6-[(2-hydroxyethyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-[(5-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1,2,4-oxadiazol-3-yl)methyl]morpholine
9-(3-chlorobenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]butan-1-one
2-({7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)-4-methoxyphenol
(3S,4R)-3-benzyl-4-methyl-1-(2-methylpyrimidine-5-carbonyl)piperidin-4-ol
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(pyridin-4-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-N-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-amine
1-(5-propyl-1,3,4-oxadiazol-2-yl)-3-(pyrrolidine-1-carbonyl)piperidine
4-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]pyridine
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-(3-hydroxy-3-methylbutyl)benzamide
1-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}piperidin-4-amine
3-({[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
3-chloro-5-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-(thiolan-3-yl)piperidin-4-amine
N,N-dimethyl-7-(oxane-4-carbonyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,5R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2,6-dihydroxy-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}benzamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
methyl 3-{[4-(dimethylamino)phenyl]methyl}-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-ethyl-N-methylpyrimidin-4-amine
(4aS,7aR)-1-[(3-fluoro-2,4-dimethylphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(4-fluorophenyl)ethyl]-N-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
methyl 4-{[(2-{1-[1-(4-chlorophenyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
3-[(3-fluorophenyl)methyl]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-[3-(3-methoxybenzoyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
N-(1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
(5S,9aS,9bS)-2-methyl-5-[3-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-methyl-N-{[1-(3-methylbutyl)piperidin-4-yl]methyl}-1H-imidazole-4-sulfonamide
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
(1-benzothiophen-2-ylmethyl)(methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]ethan-1-one
3-(6-methoxynaphthalene-2-carbonyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine
N-({1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
1-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one