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1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-(pyridine-3-carbonyl)-1,4-diazepan-2-one
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-{[(2-hydroxyethyl)(propan-2-yl)amino]methyl}benzamide
2-amino-N-[2-(ethanesulfonyl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[(6-methylpyridin-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
1-methyl-4-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)piperidin-4-ol
5-(3-chloro-4-fluorophenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(morpholin-4-yl)pyridine-3-carboxamide
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(6-methoxyhexanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-5-(3,5-dimethylbenzoyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(furan-2-carbonyl)pyrrolidin-3-yl]methanol
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-2-methyl-5-propylpyrimidin-4-amine
3-({1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidin-4-yl}oxy)pyridine
N-benzyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
methyl 1-{4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanoyl}piperidine-2-carboxylate
5-{[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]sulfonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-3-(pyridin-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenoxy)acetamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(dimethylamino)propan-1-one
N-(1-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
4-[(2-fluorophenyl)methyl]-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidine
N-({8-[(2,4-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methoxyacetamide
5-(2-methoxyacetamido)-N-(2-methoxyethyl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidin-3-yl]methanol
(1R,7S)-N-methyl-3-[2-(4-methylphenyl)ethyl]-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-N-ethylacetamide
1-({1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azepane
4-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]pyridine-2-carboxylic acid
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyrimidin-4-yl}piperidin-4-ol
(cyclopropylmethyl)[(4-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
(2S)-2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-(methylsulfanyl)butan-1-ol
5-benzyl-3-[2-(pyrrolidin-1-yl)ethyl]-5-{1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[(3-methoxyphenyl)methyl]-4-[2-(morpholin-3-yl)acetyl]piperazin-2-one
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-(thiophen-2-ylmethyl)-1-benzofuran-2-carboxamide
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
N4-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
2-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-1,3-benzodiazole
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[(3-chlorophenyl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-cyclohexyl-N3-[2-(2-fluorophenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide