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5-(4-cyclopentylpiperazin-1-yl)-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-(3-hydroxyadamantan-1-yl)-3-[(thiophen-2-ylmethyl)amino]benzamide
(4aS,7aR)-1-(2,5-dimethylfuran-3-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[3-methyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
1-(1-benzothiophen-2-ylmethyl)-4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(2R,3R)-3-amino-1'-(5-hydroxypyrazine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4'-(cyclobutylmethyl)-1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-{1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}phenoxy)ethan-1-ol
2-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,3-thiazole
2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-propyl-1,3,4-oxadiazol-2-amine
6-chloro-N,N-dimethyl-3-({[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-propyl-3-(thiomorpholine-4-carbonyl)-5-[4-(thiophene-2-carbonyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole
2-methyl-4-(4-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}phenyl)but-3-yn-2-ol
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-methyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2E)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(pyridin-2-yl)prop-2-enamide
N-{[7-(3,5-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-methylbenzamide
1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-4-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-2-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-chloro-3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(1-{[1-(1-propylpiperidin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
5-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
5-cyclopropanecarbonyl-1'-[(4-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{[(2,3-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3-methylthiophene-2-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
{3-[(3-chlorophenyl)methyl]-1-(oxane-4-carbonyl)piperidin-3-yl}methanol
1-(3-chloropyridin-2-yl)-4-(1-methylpiperidin-4-yl)-1,4-diazepan-6-ol
5-{[4-(diethylamino)phenyl]methyl}-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[2-(cyclohex-1-en-1-yl)acetyl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
6-{2-[(4-chlorophenyl)methoxy]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[(2-chlorophenyl)methyl]-3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]propanamide
3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-2-ol
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
N-[3-(methylsulfanyl)propyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-hydroxy-1-methyl-3-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}piperidin-2-one
1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
3-hydroxy-S-[2-(3-methoxypropanoyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]butane-1-sulfonamido
1-[(1-{6-[(4-hydroxybutyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(3S,9aR)-3-benzyl-8-[(3,4-dimethylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2,3-dimethylphenyl)-2-{2-[2-(thiophen-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}acetamide
(1r,4r)-4-{[2-(dimethylamino)-2-(3-methylphenyl)acetamido]methyl}cyclohexane-1-carboxylic acid
(1-benzofuran-2-ylmethyl)(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-[(3S,4R)-1-benzyl-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-en-1-yl)amine
5-ethyl-N-(1-propylpiperidin-3-yl)pyrimidin-2-amine
9-(3-chloro-4-fluorobenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one