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3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(3-methylbutanoyl)piperidin-4-yl]oxy}benzamide
2-(4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazin-1-yl)pyridine-3-carbonitrile
3-(methoxymethyl)-1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-amino-3-(3,4-dimethoxyphenyl)propan-1-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
3-methyl-N-[3-(1,3-oxazol-5-yl)phenyl]-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(thiophen-3-yl)acetamide
2-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methoxyphenol
N-cyclopropyl-N-{[7-fluoro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-2,3-dimethoxybenzamide
3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclopentyl-N-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-[1-(1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3,5-dimethoxy-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
methyl 2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-2-oxopiperazin-1-yl)acetate
2-(2-tert-butylpyrimidin-5-yl)-N,N,7,8-tetramethylquinoline-4-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-amine
1-ethyl-4-[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]pyrrolidin-2-one
3-(3-acetylbenzoyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-methyl-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
4-(1,3-benzothiazol-2-yl)-2-{[benzyl(ethyl)amino]methyl}phenol
1-benzoyl-2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]piperidine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-2-carboxamide
3-[5-(2,4-difluorobenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]propanamide
5-phenyl-2-(pyridin-3-yl)-4-[1-(2,4,5-trifluorobenzoyl)piperidin-4-yl]pyrimidine
1-(3-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}phenyl)ethan-1-one
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-ol
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(4-methylphenoxymethyl)piperidine
1-methyl-2-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]azepane
(1S,2S)-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclohexan-1-ol
N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]-6-oxo-1-propylpiperidine-3-carboxamide
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-methyl-1,6-naphthyridine-3-carboxamide
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(4-fluorophenyl)-4-oxobutanamide
methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(4-aminopyrimidin-2-yl)-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylic acid
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-N-{[3-methyl-7-(5-methyl-1H-indole-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-phenylacetamide
3-fluoro-2-(3-methoxyphenyl)pyridine
2-methyl-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
6-[4-(3-fluorophenyl)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
9-[2-(ethylsulfanyl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-4-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}aniline
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(propane-1-sulfonyl)piperidine
N-[(3S)-1-benzylpyrrolidin-3-yl]-N,1-dimethyl-5-phenyl-1H-pyrazole-3-carboxamide
5-[3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
N-[(2,3-dimethoxyphenyl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
4-(8-methoxyquinolin-2-yl)-N,N-dimethylbenzamide