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N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(methylsulfanyl)propanoyl]pyrrolidine-3-carboxylic acid
N-[2-(2-fluorophenyl)-1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
5-[(3-methoxyphenyl)methyl]-3-methyl-5-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2,5-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,3-thiazole-4-carboxamide
N-methyl-2-(morpholin-4-yl)-N-[2-(pyridin-2-yl)ethyl]-2-(pyridin-3-yl)acetamide
8-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-3-yl)propanamide
5-(4-cyclohexylpiperazine-1-carbonyl)-2,3-dimethylbenzene-1-sulfonamide
5-[1-(2-aminoacetyl)pyrrolidin-2-yl]-N-(2-methyl-1-benzofuran-5-yl)thiophene-2-carboxamide
2-(methoxymethyl)-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine
N-[3-(5-methyl-4-{[2-(3-methylphenyl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
1-cyclohexyl-4-(3-ethynylbenzoyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-(furan-2-carbonyl)-N-(1-phenoxypropan-2-yl)piperidin-4-amine
N-[3-(cyclopentyloxy)propyl]-5,6-dimethylpyrimidin-4-amine
1-{4-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]phenyl}imidazolidin-2-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,5-thiadiazole-3-carboxamide
1-benzyl-4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-[3-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)phenoxy]acetamide
ethyl 4-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoate
2-(3-phenylpropyl)-4-[3-(1H-pyrazol-4-yl)benzoyl]morpholine
4-[(2-fluorophenyl)methyl]-1-(3-methylfuran-2-carbonyl)-1,4-diazepan-5-one
N-[2-(1-benzylpiperidin-2-yl)ethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(benzylsulfamoyl)[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]amine
N-methyl-N-[2-(methylamino)ethyl]-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
methyl 3-acetamido-1-ethyl-5-[(2-methylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-4-(1H-pyrazol-4-yl)butan-1-one
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-{1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
9-methoxy-7-(pyridin-3-yl)-4-[3-(trifluoromethyl)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[2-(4-methoxyphenoxy)acetyl]-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
7-(2-cyclohexylethyl)-2-(6-methylpyridine-2-carbonyl)-2,7-diazaspiro[4.5]decane
1-({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperidin-4-ol
N-[(3,4-dimethoxyphenyl)methyl]-4-fluoro-N-(pyridin-3-ylmethyl)benzamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]propan-1-one
2-(3,4-dimethoxyphenyl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-indole
N-[(2-methoxyphenyl)methyl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1-cyclohexyl-3-(2-fluorophenyl)-3-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
2-ethyl-1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine
6-methoxy-4-[3-(4-methoxyphenyl)propanoyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-[(3-fluorophenyl)methyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-sulfonamide
{2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
(3aR,6aR)-N-(2,3-dihydro-1H-inden-2-yl)-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
6-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-{3-[(1-hydroxyhexan-2-yl)amino]butyl}phenol
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methoxyethyl)-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole