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1-[(4-methylphenyl)methyl]-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
ethyl 4-benzyl-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxylate
{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
(1S,4S)-5-[2-(2-chlorophenyl)acetyl]-2-(3,4-difluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-phenyl-4-[2-(prop-2-yn-1-yloxy)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-methylpyrimidine
3-(4-{[3-(dimethylamino)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
N-(2-methoxyethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
propyl (2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-[2-(methylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-(5-methyl-1,3-oxazole-4-carbonyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)cyclopropanesulfonamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
1-(cyclohexylmethyl)-3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-3-phenylpyrrolidine-2,5-dione
N-{1-[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-{4-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]phenoxy}propanoic acid
1-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}-1H-pyrazole
1-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
2,2-diphenyl-N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
(2S,4R)-N-ethyl-4-[3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propanamido]-1-methylpyrrolidine-2-carboxamide
1-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
{1-[(5-ethylfuran-2-yl)methyl]-3-(3-phenylpropyl)piperidin-3-yl}methanol
(3aS,6aS)-2-(2-hydroxyethyl)-5-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}piperidin-4-amine
N-[(3R,4S)-4-propyl-1-(1H-1,2,3-triazole-5-carbonyl)pyrrolidin-3-yl]methanesulfonamide
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]pyridin-2-amine
1-(1H-indol-2-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(furan-2-carbonyl)-1,4-diazepane
2-[(3S,4R)-4-amino-1-(2,3-dimethyl-1H-indole-7-carbonyl)pyrrolidin-3-yl]ethan-1-ol
1-{4-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonane-7-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-{2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-oxoethyl}methanesulfonamide
2-(4-fluorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
2-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)azetidin-3-yl]pyridine
1-[3-(3-chlorophenyl)phenyl]-3-[3-(3-hydroxypiperidin-1-yl)propyl]urea
N-[1-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]-2-methoxyacetamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-amine
[(1-ethylpiperidin-3-yl)methyl](methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
2-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}-N-[(2-fluorophenyl)methyl]acetamide
3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(6-methylpyridine-3-carbonyl)piperidine-4-carboxamide
1-methoxy-8-{[4-(propan-2-yloxy)phenyl]methyl}-1,8-diazaspiro[4.5]decan-2-one
7-(3,4-dimethoxyphenyl)-9-methoxy-4-[(2-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-3-benzyl-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(benzyloxy)-8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1,8-diazaspiro[4.5]decan-2-one
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one