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2-[(1E)-3,3-dimethylbut-1-en-1-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-methoxypiperidine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(3-hydroxypiperidin-1-yl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
6-(2-fluorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{2-[({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)amino]ethyl}piperidin-2-one
2-amino-3-ethyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
4-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-oxazepan-6-ol
5-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
3-cyclohexyl-N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(cyclohexylmethyl)-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-2,1-benzoxazole-3-carboxamide
1-(cyclopropylmethyl)-4-(2-fluoro-4-methylbenzoyl)-2-(propan-2-yl)-1,4-diazepane
4-(2,5-dimethoxybenzoyl)-N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
1-(azocan-1-yl)-2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]ethan-1-one
6-(2-ethylpiperidine-1-carbonyl)-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole
2-(2-methyl-1,3-thiazol-4-yl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]acetamide
2-methyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
[2-(3,5-dimethylphenoxy)ethyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2,5-difluoro-N-[1-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
1-(4-methoxyphenyl)-6,6-dimethyl-4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-2-one
2-amino-N-cyclopropyl-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(4-ethylphenyl)methyl]acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(morpholin-4-yl)propanamide
(4-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}phenyl)methanol
5-methyl-N-[2-(pyridin-4-yl)ethyl]-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-(5-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}thiophen-2-yl)prop-2-yn-1-ol
4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
2-{4-[5-(3-methoxyphenyl)furan-2-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
N-cyclopentyl-1-methyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
{1-[(3,4-dimethoxyphenyl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-(3,4-dimethylphenyl)-2-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
2-(methylsulfanyl)-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
N-(5-methyl-4H-1,2,4-triazol-3-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carboxamide
5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-ethoxy-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-({7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
2-{[1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]oxy}pyrimidine
3,3-dimethyl-1-[(5-{[3-(propan-2-yloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
4-{1-[1-(dimethylcarbamoyl)piperidine-4-carbonyl]piperidin-3-yl}benzoic acid
3-methyl-7-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-2-cyclopentyl-N-(2-methoxyethyl)acetamide
7-acetamido-N-[1-(naphthalen-1-yl)ethyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-amine
(2R,3R)-3-amino-1'-(5-chloro-2-methylbenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-({[2-(azocan-1-yl)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
5-[({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-[2-(pyridin-3-yloxy)ethyl]propanamide