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ethyl[(5-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]methylamine
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(5-chloro-2-methoxybenzoyl)piperidine
1-(2-methyl-1,3-thiazole-5-carbonyl)-4-(2-phenoxyethyl)piperazine
methyl 4-{2-[benzyl(methyl)carbamoyl]ethyl}piperidine-1-carboxylate
N,1-dimethyl-5-({[1-(piperidin-1-yl)cyclopentyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(2-methoxyacetyl)-N-(2-methylquinolin-8-yl)-1,4-diazepane-1-carboxamide
5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
(2S)-2-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}-4-(methylsulfanyl)butan-1-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(4-fluorophenyl)ethyl]piperidine-3-carboxamide
2-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
4-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
2-[(1S,5R)-3-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
{1-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]pentan-2-yl}dimethylamine
4-{[6-(4-methoxy-3-methylphenyl)pyridin-3-yl]methyl}morpholine
8-[(2,6-dimethoxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-2-(4-methyl-1,4-diazepane-1-carbonyl)pyrrolidin-1-yl]methyl}phenol
(1R,2R,4R)-N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyridin-3-ylmethyl)piperazine
6-(1,4-oxazepan-4-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}benzamide
1-[(1S,5R)-6-[2-(1H-imidazol-2-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5-propyl-1-benzofuran-2-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)acetamide
5-phenyl-N-[4-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]pentanamide
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(5-methylpyrimidin-2-yl)amino]-3-(piperidin-1-yl)propan-2-ol
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methanol
(3R,5S)-N-(4-fluorophenyl)-1-(1H-indol-3-ylmethyl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
1-(2-{[2-(3,4-dimethylphenoxy)ethyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,3-dimethylbutanamide
5-(methoxymethyl)-3-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
1-cyclopentyl-N-[(4-fluorophenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(1H-indazol-1-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
N-[(2R,3R)-2-methoxy-1'-(thian-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
(3R,4R)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-(quinolin-2-ylmethyl)piperidin-3-ol
3-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1-(oxan-4-yl)urea
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine
2-(1H-indol-3-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
4-(2-methyl-1,3-thiazole-4-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
2-[methyl(2-phenylethyl)amino]-N-propyl-2,3-dihydro-1H-indene-2-carboxamide
3-[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-fluorobenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-(furan-2-ylmethyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(prop-2-en-1-yl)acetamide
1-[5-methoxy-2-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(2S)-2-amino-1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
1-(2-{[(1-methyl-1H-pyrazol-4-yl)carbamoyl]amino}ethyl)piperidine-3-carboxamide