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4-{5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}-1,4-oxazepane
4-[5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-(quinolin-6-yloxy)piperidine-4-carboxamide
5-(2-methoxy-3-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(4aR,7aS)-1-ethyl-4-[(3-phenylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine-4-carboxamide
3-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
2-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
(4aR,8aS)-6-(4-methoxybenzoyl)-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-hydroxy-N-[(3R,4S)-4-(propan-2-yl)-1-[(3,4,5-trifluorophenyl)methyl]pyrrolidin-3-yl]propanamide
8-(2-methylquinolin-4-yl)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,8-diazaspiro[4.5]decane
N-ethyl-3-(2-methoxyphenyl)-N-(pyridin-4-ylmethyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
methyl 3-(cyclobutylmethoxy)-5-{[1-methyl-1-(methylcarbamoyl)ethyl]carbamoyl}benzoate
N-(1-methylpiperidin-4-yl)-2-oxo-N-(2-phenylethyl)-1,2-dihydroquinoline-3-carboxamide
1-{2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]acetyl}-N,N-diethylpiperidine-3-carboxamide
1-ethyl-N-(9H-fluoren-9-yl)-2-oxo-1,2-dihydropyridine-4-carboxamide
N-(3,4-difluorophenyl)-6-(dimethyl-1,3-thiazole-5-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
5-(methoxymethyl)-N-[(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-2-carboxamide
(2S)-2-acetamido-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-methylpentanamide
4-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholin-4-yl)-6-(propan-2-yl)pyrimidin-2-amine
1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]urea
2-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methylpyrimidine-5-carboxamide
1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}piperidine-3-carboxylic acid
[4-({[(5-chlorothiophen-2-yl)methyl](methyl)amino}methyl)oxan-4-yl]methanol
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
5-methyl-1-(4-{4-[(1-methyl-2-oxopyrrolidin-3-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
2-({1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidin-4-yl}formamido)acetamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
1-(2,4,6-trimethyl-3-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-one
N-[4-(2H-1,3-benzodioxol-4-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]methanesulfonamide
2-({3-[3-(6-methylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}methyl)quinoline
7-(4-chloro-1H-pyrazole-3-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(pyrazin-2-yl)ethyl]amine
(2S,4R)-4-amino-N,N-diethyl-1-(pyridine-3-sulfonyl)pyrrolidine-2-carboxamide
2-[benzyl(methyl)amino]-N-[1-(pyrazin-2-yl)propan-2-yl]-2,3-dihydro-1H-indene-2-carboxamide
1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
(heptan-4-yl)[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amine
4-[1-(2-ethoxy-2-methylpropanoyl)piperidin-3-yl]benzoic acid
N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-6-carboxamide
2-methyl-N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
ethyl 4-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]quinoline-3-carboxylate
N-[2-(1,2,3-thiadiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
2-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole