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7-fluoro-2-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}quinoline-4-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
1-(benzyloxy)-8-(2-fluorobenzoyl)-1,8-diazaspiro[4.5]decan-2-one
3-(2-fluorophenyl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-phenylpropan-1-one
2-{[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}ethan-1-ol
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
N-(2-methoxyethyl)-5-(5-methoxypyridin-3-yl)furan-2-carboxamide
N-(2,4-dimethoxyphenyl)-3-[1-(pyridine-4-carbonyl)piperidin-4-yl]propanamide
1-ethyl-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)propanamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-amino-4-propyl-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
(3R,4R)-1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-4-(hydroxymethyl)piperidin-3-ol
1-[(4-{furo[3,2-c]pyridin-4-yloxy}-3-methylphenyl)methyl]pyrrolidine
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4-oxo-1,4-dihydroquinoline-2-carboxamide
2-fluoro-N-(4-{4-[(pyridin-4-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
6-(1H-pyrazole-4-carbonyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-1-phenyl-1H-1,2,3,4-tetrazole
9-benzoyl-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-ethyl-1-(2-phenylethyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-(furan-2-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-(9H-purin-6-yl)piperidin-4-amine
N-cyclopropyl-4-(3-fluorophenyl)-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}benzamide
1-methyl-5-phenyl-N-[3-(pyrrolidin-1-yl)propyl]-1H-pyrazole-3-carboxamide
1-[(2,3-difluoro-4-methoxyphenyl)methyl]-4-[(4-fluorophenyl)methyl]-1,4-diazepane
(4aR,8aS)-1-[2-(2-fluorophenyl)ethyl]-6-{[2-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-chloropyridin-4-yl)methyl]piperidin-3-ol
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-(methylsulfanyl)acetamide
1-[1-(piperidin-4-ylmethyl)piperidin-4-yl]butan-1-one
2-(4-amino-3-methoxyphenyl)-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
7-[(3-methylphenyl)methyl]-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}(methyl){[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-(2-methoxyethyl)-6-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}piperidine-3-carboxamide
(3S,4S)-1-(4-aminopyrimidin-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
3-[(4-fluorophenyl)methyl]-N-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
1-(6-aminopyrimidin-4-yl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
5,8-dimethyl-2-(morpholin-4-ylmethyl)quinolin-4-ol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N,2,6-trimethylquinoline-3-carboxamide
({5-[1-(1H-indole-2-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(pyridin-4-yl)-5-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrimidin-4-ol
1-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carbonitrile
5-{[2-(2-ethyl-1-benzofuran-3-yl)-1H-imidazol-1-yl]methyl}-3-methyl-1,2-oxazole
2-ethyl-6-(3-methoxy-2-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
6-(2,3-dimethoxybenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-methyl-N-[2-(morpholin-4-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one