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3-(dimethylamino)-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-(pyridine-4-carbonyl)piperidine-2-carboxamide
5-[2-(benzylamino)ethyl]-1-[(3-chlorophenyl)methyl]pyrrolidin-2-one
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methylphenyl)acetamide
1-methyl-2-{[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-1,3-benzodiazole
N-[(2R,3R)-2-ethoxy-1'-(1H-indol-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[(2R,3R)-1'-[(2,5-dimethoxyphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-ethyl-4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-1-(propan-2-yl)piperazine
3-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-1-(5-methanesulfonyl-2-methylphenyl)-3-methylurea
N-[(2R,3R)-1'-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
N-(4-fluorophenyl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperazine-2-carboxamide
N'1-[(1-cyclopentylpiperidin-4-yl)methyl]-N'1-(pyridin-3-ylmethyl)cyclopropane-1,1-dicarboxamide
3-[2-(2-methylpropanesulfonyl)ethyl]-1-(1-phenyl-1H-pyrazol-5-yl)urea
4-[5-(3-chlorothiophene-2-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
5-{1-[(2E)-3-(2,6-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
3-(1H-1,2,4-triazol-3-yl)-1-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]urea
6-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
7-(2-butoxy-5-methylphenyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
2-(2,4-difluorophenoxy)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)ethan-1-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
6-ethoxy-4-methyl-2-{4-[4-(pyridin-3-yloxy)piperidin-1-yl]azepan-1-yl}quinazoline
5-{[2-methyl-4-(pyrimidin-4-yl)piperazin-1-yl]sulfonyl}isoquinoline
2-[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(5-methylpyridin-2-yl)acetamide
2-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
1-ethyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-3-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
1-(3-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(3-methylthiophen-2-yl)ethyl]acetamide
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-2-one
5-ethyl-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-1,2-oxazole-3-carboxamide
9-[(2R)-2-aminopropanoyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
2-(furan-2-yl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]azepane
3-[1-(2-methyl-1,3-benzothiazole-6-carbonyl)piperidin-3-yl]benzoic acid
N-[1-(4-fluorophenyl)propyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[2-methoxy-4-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)phenoxy]acetamide
methyl 3-acetamido-1-methyl-5-[(naphthalen-1-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-methoxy-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
5-methyl-N4-{[3-(trifluoromethoxy)phenyl]methyl}pyrimidine-2,4-diamine
N-[2-(3-methoxyphenyl)ethyl]-6-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methylpropanamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(morpholin-4-yl)butan-1-one
(1R,7S)-6-[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(2-methoxy-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2,2-dimethylpropyl)-4-phenyl-1H-imidazole