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5-methyl-2-(naphthalen-2-yl)-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
6-(methoxymethyl)-N,1-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-(1,2-oxazol-3-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(oxan-2-ylmethyl)propanamide
N-[2-benzyl-7-(4-hydroxypiperidine-1-carbonyl)-1-methyl-1H-1,3-benzodiazol-5-yl]propanamide
6-[2-(1-methylpyrrolidin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(4-{4-[methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]piperidin-1-yl}benzoyl)piperidin-3-ol
N-(3-chloro-4-methoxyphenyl)-6-(3,5-dimethoxybenzoyl)-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-9-[(2-methyl-2H-1,2,3-benzotriazol-4-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-(1-{7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carboxamide
3-{5-[2-(phenylsulfanyl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
8-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3,4-dimethoxyphenyl)methyl]-2-methoxy-N-(pyridin-4-ylmethyl)benzamide
1-(2-oxo-2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-ethyl-3-methylpiperidine-1-carbonyl)-6-methyl-4H-pyran-4-one
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-1-yl)-4H-1,2,4-triazole
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3-chloro-4-fluorophenyl)-N'-[(1r,4r)-4-hydroxycyclohexyl]propanediamide
N-[2-(3-chlorophenoxy)ethyl]-N-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-methyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-N-(propan-2-yl)acetamide
2-{[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
(3R)-3-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinoline
N-[3-(1H-imidazol-1-yl)butyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
6-methyl-2-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}methyl)quinolin-4-ol
1-{4-[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]piperidin-1-yl}ethan-1-one
1-[(3-fluorophenyl)methyl]-4-(1H-imidazol-2-ylmethyl)piperazin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,7-trimethyl-1H-indole-2-carboxamide
3-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3,5-difluoro-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]pyridine-2-carboxamide
methyl 1-[(4-amino-6-methylquinazolin-2-yl)methyl]piperidine-2-carboxylate
(2E)-N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3,4-dimethoxyphenyl)prop-2-enamide
methyl 5-[2-(4-fluorophenyl)morpholine-4-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylate
1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
3-[5-(1H-indol-2-yl)-1,3,4-oxadiazol-2-yl]-1-(1,2-oxazinan-2-yl)propan-1-one
1-{5-methoxy-2-[({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]phenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-fluoro-2-methoxyphenyl)-3-(piperidine-1-carbonyl)pyridine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-4-(trifluoromethyl)benzamide
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-N-(2,4-dimethoxyphenyl)propanamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-{[2-(pyridin-4-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2E)-3-(3,4-difluorophenyl)-N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)prop-2-enamide