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{5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-imidazol-2-yl]furan-2-yl}methanol
N-({7-[(2E)-3-(4-chlorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)propanamide
ethyl 2-{1-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidin-4-yl]-N-methylformamido}acetate
5-[4-(aminomethyl)piperidin-1-yl]-2-(pyridin-4-ylmethyl)-2,3-dihydropyridazin-3-one
[(3,4-dimethoxyphenyl)methyl](methyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
ethyl 4-(2-phenoxyethyl)-1-(3-phenylprop-2-ynoyl)piperidine-4-carboxylate
6-(azepan-1-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
[(2S)-1-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}pyrrolidin-2-yl]methanol
5-butyl-1-(2-methoxyphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
2-[(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)methyl]benzonitrile
2-amino-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-6-(propan-2-yl)pyrimidine-4-carboxamide
N-ethyl-2-{4-[8-(trifluoromethyl)quinolin-4-yl]piperazin-1-yl}acetamide
1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-4-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-2-one
ethyl 4-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
4-[3-(4-chlorophenyl)-3-phenylpropanoyl]piperazin-2-one
methyl 3-benzamido-1-(furan-2-ylmethyl)-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(pyrazin-2-yl)ethyl]benzamide
N-ethyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
5-(2-chlorophenyl)-4-[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]pyrimidine
ethyl 4-{3-[(3-phenylpropanamido)methyl]piperidin-1-yl}piperidine-1-carboxylate
N-[1-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)propan-2-yl]-2-(phenylsulfanyl)acetamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-yl]propan-1-ol
1-[(4-methylphenyl)methyl]-4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
1-[(3-methoxyphenyl)methyl]-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
5-[4-(2-chlorophenyl)-3-oxopiperazine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-phenyl-1H-pyrazole-5-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]pyrrolidine-2-carboxamide
1-{4-[2-(3,4-dichlorophenyl)morpholin-4-yl]piperidin-1-yl}ethan-1-one
7-methoxy-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1,2,3,4-tetrahydronaphthalen-2-amine
(4aS,8aS)-2-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-decahydroisoquinolin-4a-ol
4-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
1-methyl-N-[(3-methylpyridin-4-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-(cyclopropylmethyl)-1-methyl-4-(2-methylpyridin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[3-({[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amino}methyl)phenyl]ethan-1-one
N,N-dimethyl-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-sulfonamide
(1R,5R)-6-[(4-cyanophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
N-methyl-4-oxo-1-(2-phenylethyl)-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzamide
2-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
6-(cyclohex-3-en-1-ylmethyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-[(3-fluorophenyl)methyl]-3-{[3-(2-hydroxyethoxy)phenyl]methyl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(2-hydroxyethyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-benzyl-3-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-N-methylpropanamide
3-({2-[methyl(2-phenylethyl)amino]ethyl}carbamoyl)benzoic acid
7-(2-methoxyethyl)-2-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one