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1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
methyl 4-(2-phenyl-1H-imidazol-1-yl)butanoate
(2R,3R)-1'-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(2-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
6-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-hydroxyethyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
4-benzyl-3-ethyl-1-{thieno[2,3-d]pyrimidin-4-yl}-1,4-diazepan-5-one
1-cyclopentyl-4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
ethyl 2-(4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}morpholin-3-yl)acetate
4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(trifluoromethyl)morpholine
N-({1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)acetamide
2-(4-{[4-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
1-(2-cyclohexylethyl)-N-[2-(4-fluorophenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-ethoxy-5-[3-(1H-pyrazol-3-yl)phenyl]benzamide
N-[(3-methylphenyl)methyl]-3-(piperidine-1-carbonyl)-N-(propan-2-yl)pyrazine-2-carboxamide
1-methyl-3-(2-methylpropyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
(3E)-2-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}hept-3-enoic acid
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetic acid
5-(naphthalen-2-ylmethyl)-5-(3-oxo-3-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}propyl)pyrrolidin-2-one
4-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
6-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
6-{1-[2-(1H-imidazol-5-yl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl}pyridin-2-amine
4-oxo-5-phenoxy-1-[1-(pyridin-2-yl)propyl]-1,4-dihydropyridine-3-carboxylic acid
4-hydroxy-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
methyl (2S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
N-cyclopropyl-1-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-[2-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
8-[(2,4-dimethoxyphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-benzyl-1-(2-hydroxyethyl)-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
2-methyl-4-(4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}phenyl)butan-2-ol
4-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine
9-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-benzyl-4-(5-methylpyrazine-2-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-(4-{[3-(dimethylamino)propyl](methyl)amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(3-methylbenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-ethyl-4-{[3-oxo-4-(2-phenylphenyl)piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[3-({[2-(azepan-1-yl)ethyl](ethyl)carbamoyl}amino)-4-methoxyphenyl]acetamide
N-[(2R,3R)-1'-(1H-indole-6-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
2-butanoyl-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-[(3,4-dimethylphenyl)amino]-N-(4H-1,2,4-triazol-4-yl)cyclohexane-1-carboxamide
N,N-diethyl-5-(pyridin-4-yl)furan-2-carboxamide
1-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
N-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-propylpyrrolidin-3-yl]-3-methanesulfonylpropanamide
7-methyl-2-[2-(propan-2-yl)pyrimidine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-(pyrazin-2-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-(butan-2-yl)-3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-methyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1,3-thiazole-4-carboxamide