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2-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
3-(azepane-1-sulfonyl)-5-(pyrimidin-5-yl)benzoic acid
3-{5-[1-(2-ethoxyacetyl)piperidine-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(1S,2R)-N2-tert-butyl-N1-methyl-N1-[(3-methylthiophen-2-yl)methyl]cyclohexane-1,2-dicarboxamide
N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
9-(2-methoxypropanoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-(3-chlorobenzoyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-methoxy-4-methyl-1,3-thiazole-5-carboxamide
1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
5-[1-(benzylcarbamoyl)-6-azaspiro[2.5]octane-6-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
N-({8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
4-methyl-2-(4-methylpiperazin-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyrimidine-5-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-6-methylpyridine-3-carboxamide
N-(1-{7-[2-(3,4-dimethoxyphenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-(dimethylamino)acetamide
N-(diphenylmethyl)-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-(1-methoxypropan-2-yl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-(isoquinolin-5-ylmethyl)-N,4-dimethyl-1,2,3-thiadiazole-5-carboxamide
(2-methoxyethyl)[(2-methyl-2H-indazol-3-yl)methyl][(4-methylphenyl)methyl]amine
1-(4-{[(3-chloro-1-benzothiophen-2-yl)methyl](methyl)amino}piperidin-1-yl)ethan-1-one
N-{[8-(6-hydroxypyridine-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
4-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)-1,2-dihydroisoquinolin-1-one
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2-[(2-methylphenyl)sulfanyl]acetamide
N-cyclobutyl-2-[2-(diethylamino)acetyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(methylsulfanyl)propan-1-one
methyl 3-{4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl}propanoate
N-[(2-amino-1,3-thiazol-4-yl)methyl]-4-ethoxypyrimidin-2-amine
(2S)-2-amino-3-hydroxy-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
4-(1H-imidazol-1-yl)-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
3-(4-fluoro-2-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
{3-[(2-fluorophenyl)methyl]-1-(quinolin-2-yl)piperidin-3-yl}methanol
N-cyclopentyl-N-{[3-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
4-{[(3-acetylphenyl)methyl]amino}-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
2-(4-{2-[(2-methoxyphenyl)methoxy]phenyl}-3,5-dimethyl-1H-pyrazol-1-yl)acetamide
4-(3,5-dimethyl-1H-indol-2-yl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{2-[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3-oxazinan-2-one
(1S,6R)-9-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonane
2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propane-1,3-diol
ethyl 5-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
ethyl 1-methyl-5-[(2-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-hydroxy-1-(2-phenylethyl)-3-({[2-(1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)piperidin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazole
4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridin-2-amine
(1S,5R)-3-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-fluorophenoxymethyl)-1-(3-methyl-1H-pyrazole-4-carbonyl)piperidine
3-ethyl-1-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)urea
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
5-[(2-fluorophenyl)methyl]-3-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
ethyl 4-(6-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(4-methylpiperidin-1-yl)ethan-1-one