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1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
N-(2H-1,3-benzodioxol-5-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-amine
1-(3-methylbutyl)-8-[3-(5-methylfuran-2-yl)butyl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-phenyl-1H-pyrrole-2-carboxamide
6-[(diethylamino)methyl]-N-(2,2-dimethyloxan-4-yl)-N-ethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-benzyl-1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-({3-methyl-7-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
3-[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]propane-1,2-diol
5-{2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
ethyl 2-{[5-(7-hydroxy-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)pyrimidin-2-yl]amino}acetate
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[(4-fluorophenyl)methyl]piperidine
(2E)-1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-phenylprop-2-en-1-one
3-[(4-methoxyphenyl)methyl]-4-(4-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-fluorophenyl)-N-[(1-hydroxycyclohexyl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
9-hydroxy-3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
ethyl 1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-[1-(2-methoxyethyl)-1H-indol-3-yl]pyridine-3-carbonitrile
1-{2-[methyl({[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amino]ethyl}piperidin-2-one
N5-cyclooctyl-1-(2-methoxyethyl)-N3-methyl-4-oxo-N3-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(2-fluorophenyl)-3-phenyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-{8-[2-(3-chloro-5-fluorophenyl)acetyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
5-[2-(methylsulfanyl)-1,3-thiazol-4-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-2-(3-methylphenyl)pyrimidine
4-(4-methanesulfonylpiperazine-1-carbonyl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
N-cyclopentyl-4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
2-amino-4-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-6-(thiophen-3-yl)pyridine-3-carbonitrile
1-(propane-1-sulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1H-indol-5-yl)-4-(pyrrolidine-1-sulfonyl)piperazine-1-carboxamide
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]benzoic acid
3-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}quinoline
4-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-2,1,3-benzoxadiazole
3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1-methyl-1-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
3-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)-N-(1-phenylcyclopropyl)propanamide
1,4-dimethyl-9-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-1,4,9-triazaspiro[5.5]undecane
(4aS,7aR)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclopropyl-N-[2-(2-fluorophenoxy)ethyl]-6-oxopiperidine-3-carboxamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
1-{2-[2-(1H-indol-3-yl)acetamido]ethyl}-N-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-methoxybenzoic acid
2-({[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-methyl-1H-pyrazole-5-carboxamide
7-(cyclobutylmethyl)-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridin-2-amine
3,3,3-trifluoro-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
7-methyl-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
1,9-dimethyl-4-(5-propylthiophene-3-carbonyl)-1,4,9-triazaspiro[5.5]undecane
N-{2-[methyl(phenyl)amino]ethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide