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2-(5-{6-methylimidazo[2,1-b][1,3]thiazol-3-yl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)pyridine
5-cyclopentyl-3-({3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,2,4-oxadiazole
1-methyl-3-(3-phenylphenyl)-6-[3-(pyridin-2-yl)propanoyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
9-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,9S)-5-amino-3-[3-(2-hydroxyethoxy)phenyl]-13-methyl-6,13-diazatricyclo[7.3.1.02,7]trideca-2,4,6-triene-4-carbonitrile
methyl 1-{2-hydroxy-3-[3-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
8-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[1-(adamantan-1-yl)propan-2-yl]-3,4-dihydropteridin-4-one
2-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridine-3-carboxamide
4-[1-cyclohexyl-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]butanamide
2-{1-[(1-cyclopentylpiperidin-4-yl)methyl]-1H-imidazol-2-yl}pyridine
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-(oxan-4-yl)-4-phenyl-1H-imidazole
methyl[2-(morpholin-4-yl)ethyl]{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(1H-pyrazole-3-carbonyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-acetyl-N-[(3S,4R)-4-ethoxyoxolan-3-yl]thiophene-3-carboxamide
N-cyclopropyl-5-(6-methoxypyridin-3-yl)thiophene-2-carboxamide
N4-methyl-N6-(propan-2-yl)-N4-(pyridin-3-ylmethyl)pyrimidine-2,4,6-triamine
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-N-[2-(1,3-thiazol-2-yl)ethyl]pyrimidin-2-amine
N-cyclooctyl-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
{1-[2-(morpholin-4-yl)-6-phenylpyridine-3-carbonyl]piperidin-4-yl}diphenylmethanol
3-(aminomethyl)-4-[4-chloro-3-(trifluoromethyl)phenyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(3-aminopropyl)-1H-1,2,3-triazole-4-carbonyl]-N-(4-methoxyphenyl)piperidin-3-amine
1-(6-aminopyrimidin-4-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-6-carboxylic acid
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(furan-3-ylmethyl)-N-methylpropanamide
8-fluoro-2-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}quinoline
N-{4-[2-(hydroxymethyl)pyridin-4-yl]phenyl}methanesulfonamide
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3R,5S)-N-[(2,5-dimethylphenyl)methyl]-1-(pyridin-3-ylmethyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
2-(ethylamino)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}pyrimidine-5-carboxamide
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
4-methyl-5-(3-phenylpiperazine-1-carbonyl)-2-(propan-2-yl)pyrimidine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(4-hydroxyphenyl)methyl]piperidine-4-carboxylic acid
3-amino-N-[3-methyl-1-(4-methylquinolin-2-yl)-1H-pyrazol-5-yl]piperidine-1-carboxamide
2-[2-(hydroxymethyl)pyridin-4-yl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]-2-(trifluoromethyl)morpholine
7-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-methyl-1-[(1-methylpiperidin-3-yl)methyl]-1,4-dihydroquinolin-4-one
(2S,4S,5R)-5-(4-chlorophenyl)-4-{[2-(1H-imidazol-4-yl)ethyl]carbamoyl}-1,2-dimethylpyrrolidine-2-carboxylic acid
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
6-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-(2-methylphenyl)-3-{1-[1-(4,4,4-trifluorobutan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-[4-(oxane-4-carbonyl)piperazin-1-yl]-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
9-(3-hydroxy-2-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-ethyl-3-(2-methylpropyl)-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-pyrazole-5-carboxamide
N-[2-(2-fluorophenyl)-1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-fluoro-4-methylbenzoyl)pyrrolidine-3-carboxylic acid
ethyl 1-(6-methylpyridine-2-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate