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4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-(3-methoxypropyl)-8-(trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-butyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-2-one
(4aR,8aS)-6-(2,3-dihydro-1H-inden-2-yl)-1-[2-(2-methoxyphenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{1-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
1-ethyl-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(2-ethoxyphenyl)methyl]piperazin-2-one
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
7,7-dimethyl-2-[2-(pyrrolidin-1-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2R,3R)-3-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
1-(2-chlorophenyl)-4-{3-[methyl(1-methylpyrrolidin-3-yl)amino]propanoyl}piperazin-2-one
5-(2,4-difluorophenoxymethyl)-N-(1-methoxybutan-2-yl)-1,2-oxazole-3-carboxamide
2-(2,5-dimethylphenyl)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-[(2,6-dimethoxyphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyrimidin-4-amine
2,4-dioxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-benzylpiperidin-1-yl)-3-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]propan-1-one
1-[3-(diethylamino)pyrrolidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
2-[(2-chlorophenyl)methyl]-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]morpholine
[3-({[(5-methoxy-1,3-benzoxazol-2-yl)methyl]amino}methyl)-2,4,6-trimethylphenyl]methanol
6-(methoxymethyl)-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-(1-ethyl-1H-imidazol-2-yl)piperidine
7-(5-chloro-2-methoxyphenyl)-9-methoxy-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopentyl-5-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclopropyl-4-hydroxy-2-(3-methylphenyl)-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
4,6-dimethoxy-2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]pyrazine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(2-fluorophenyl)methyl]-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
N-ethyl-6-methyl-4-[2-(methylsulfanyl)ethyl]-2-oxo-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2R,3R)-3-amino-1'-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
diethyl({2-[2-(pyridin-2-yl)-1H-imidazol-1-yl]ethyl})amine
2-benzyl-8-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-3-acetamido-N,4-bis(4-methylphenyl)pyrrolidine-1-carboxamide
2-{3-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}acetamide
2-[2-(ethylamino)pyrimidin-5-yl]-7-fluoro-N-(1-methyl-2-oxopyrrolidin-3-yl)quinoline-4-carboxamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-cyclopropyl-3-(5-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
N-cyclohexyl-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-(prop-2-yn-1-yl)acetamide
7-(cyclobutylmethyl)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-[4-(benzyloxy)butyl]pyridine-3-carboxamide
4-fluoro-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
2-({4-[2-(2,5-dimethyl-1H-pyrrol-1-yl)ethyl]piperazin-1-yl}methyl)pyridine-3-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-(3-hydroxyquinoxalin-2-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}propanamide